Current Topics

Metalated Alkoxy Allenes as Building Blocks for Synthesis of Heterocycles

Publications

F. Cumine, A. Young, H.-U. Reißig, T. Tutttle*, J. A. Murphy*
A Computational Study of Anionic Alkoxide-Allene and Amide-Allene Cyclizations
Eur. J. Chem. 2017, 6867 – 6871.
S. Schoder, S. Kord Daoroun Kalai, H.-U. Reißig*
Novel Alkoxy-Substituted Dipyrromethenes and Near-IR BODIPY Dyes – Preparation and Photophysical Properties
Chem. Eur. J. 2017, 23, 12527 – 112533.
H.-U. Reißig*, R. Zimmer*
Cyclizations of Alkoxyallenes: Mechanisms, Intermediates, Products – A Personal Account on Solved and Unsolved Problems with Unique Allene Building Blocks
Synthesis strong>2017, 49, 3291 – 3302.
D. Gladow, S. Senf, J. Wiecko, D. Lentz, R. Zimmer, H.-U. Reißig*
New Trifluoromethyl-Substituted Heterocycles by Multicomponent Reactions of Siloxycyclopropanes
Chem. Heterocycl. Compd. 2017, 53, 416 – 421.
M. Medvecký, I. Linder, L. Schefzig, H.-U. Reißig*, R. Zimmer*
Iodination of Carbohydrate-Derived 1,2-Oxazines to Enantiopure 5-Iodo-3,6-dihydro-2H-1,2-oxazines and Subsequent Palladium-Catalyzed Cross-Coupling Reactions
Beilstein J. Org. Chem. 2016, 12, 2898 – 2905.
R. Klemme, C. Bentz, T. Zukowski, L. Schefzig, D. Lentz, H.-U. Reißig,* R. Zimmer*
Percarboxylic Acid Oxidation of α-Hydroxy-Substituted Alkoxy-allenes: The Unexpected Formation of Acyloxy-Substituted 1,2-Diketones and the Synthesis of Functionalized Quinoxalines
Synthesis 2016, 48, 1491 – 1501.
M. Wilsdorf, H.-U. Reißig*
Model Studies towards New Functionalized Bisbenzannulated [5,6]-Spiroketals
Eur. J. Org. Chem. 2016, 1555–1561.
M. Jasiński*, G. Utecht, A. Fruziński, H.-U. Reißig
Three-Step Synthesis of 3-Aminoseptanoside Derivatives Using Lithiated Methoxyallene and δ-Siloxynitrones
Synthesis 2016, 48, 893 – 905.
J. Salta, J. Dernedde, H.-U. Reißig*
Synthesis of Multivalent Carbohydrate Mimetics with Aminopolyol End Groups and their Evaluation as L-Selectin Inhibitors
Beilstein J. Org. Chem. 2015, 11, 638 – 646.
J. Salta, H.-U. Reißig*
Synthesis of Divalent Carbohydrate Mimetics by Reductive Amination with Enantiopure 1,2-Oxazines as Precursors
Synthesis 2015, 47, 1893 – 1898.
R. Zimmer, H.-U. Reißig*
Allenes in Multicomponent Synthesis of Heterocycles
in: Multicomponent Reactions in Organic Synthesis, (J. Zhu, Q. Wang, M.-X. Wang, Eds.),
WILEY-VCH, Weinheim 2015, 301 – 332.
M. Kandziora, E. Mucha, S. P. Zucker, H.-U.Reißig*
Syntheses of Mono- and Divalent C-Aminoglycosides Using 1,2-Oxazine Chemistry and Olefin Metathesis
Synlett 2015, 26, 367 – 374.
M. Kandziora, H.-U. Reißig*
Preparation of Multivalent Carbohydrate Mimetics Based on Enantiopure 1,2-Oxazines by Sonogashira Coupling and Subsequent Reductive Ring-Opening
Eur. J. Org. Chem. 2015, 370 – 377.
M. Jasiński, G. Mlostoń, M. Stolarski, W. Costa, M. Domínguez, H.-U. Reißig*
Reactions of Cycloaliphatic Thioketones and Their Oxo Analogues with Lithiated Methoxyallene: A New Approach to Vinylthiiranes
Chem. Asian J. 2014, 9, 2641 – 2648.
M. Kandziora, H.-U. Reißig*
Synthesis of Rigid p-Terphenyl-Linked Carbohydrate Mimetics
Beilstein J. Org. Chem. 2014, 10, 1749 – 1758.
R. Zimmer, H.-U. Reißig*
Alkoxyallenes as Building Blocks for Organic Synthesis
Chem. Soc. Rev. 2014, 43, 2888 – 2903.
M. K. Bera, M. Domínguez, P. Hommes, H.-U. Reißig*
The Flögel-Three-Component Reaction with Dicarboxylic Acids - An Approach to Bis(β-alkoxy-β - ketoenamides) for the Synthesis of Complex Pyridine and Pyrimidine Derivatives
Beilstein J. Org. Chem. 2014, 10, 394 – 404.

L. Bouché, M. Kandziora, H.-U. Reißig*
Synthesis of new enantiopure poly(hydroxy)aminooxepanes as building blocks for multivalent carbohydrate mimetics
Beilstein J. Org. Chem. 2014, 10, 213 – 223.

M. Jasiński, E. Moreno-Clavijo, H.-U. Reißig*
Synthesis of a Series of Enantiopure Polyhydroxylated Bicyclic N-Heterocycles from an l-Erythrose Derived Nitrone and Alkoxyallenes
Eur. J. Org. Chem. 2014, 442 – 454.

M. K. Bera, S. L. Gholap, P. Hommes, K. Neuthe, D. Trawny, J. P. Rabe, D. Lentz, R. Zimmer, H.-U. Reißig*
Synthesis and Properties of Branched Oligo(2-thienyl)- and Oligo(2,2’-bithien-5-yl)-Substituted Pyridine Derivatives
Adv. Synth. Catal. 2013, 355, 3463 – 3474.

V. M. Schmiedel, S. Stefani, H.-U. Reißig*
Stereodivergent Synthesis of Jaspine B and its Isomers using a Carbohydrate-derived Alkoxyallene as C₃-building Block
Beilstein J. Org. Chem. 2013,9, 2564 – 2569.

C. Parmeggiani, F. Cardona, L. Giusti, H.-U. Reißig*, A. Goti
Stereocomplementary Routes to Hydroxylated Nitrogen Heterocycles: Total Syntheses of Casuarine, Australine, and 7-epi-Australine
Chem. Eur. J. 2013, 19, 10595 – 10604.

S. L. Gholap, P. Hommes, K. Neuthe, H.-U. Reißig*
Per(2-thienyl)pyridines: Synthesis and Properties
Org. Lett. 2013, 15, 318 – 321.

M. Jasiński,T. Watanabe, H.-U. Reißig*
Samarium Diiodide Promoted Reduction of 3,6-Dihydro-2H-1,2-oxazines: Competition of 1,4-Amino Alcohol Formation and Ring Contraction to Pyrrole Derivatives
Eur. J. Org. Chem. 2013, 605 – 610.

T. Lechel, G. Podolan, B. Brusilowskij, C. A. Schalley, H.-U. Reißig*
Unexpected One-Step Formation of Iodo[1,3]dioxolo[4,5-c]pyridine Derivatives by a Hofmann-Löffler-Freytag Reaction: Studies on the Synthesis of a Pyridine-Containing Macrocycle
Eur. J. Org. Chem. 2012, 5685 – 5692.

M. Jasiński, Dieter Lentz, E. Moreno-Clavijo, H.-U. Reißig*
Application of L-Erythrose-Derived Nitrones in the Synthesis of Polyhydroxylated Compounds via 3,6-Dihydro-2H-1,2-oxazine Derivatives
Eur. J. Org. Chem. 2012, 3304 – 3316.
M. Jasiński, Dieter Lentz, H.-U. Reißig*
Carbohydrate-Auxiliary Assisted Preparation of Enantiopure 1,2-Oxazine Derivatives and Aminopolyols
Beilstein J. Org. Chem. 2012, 8, 662-674.
L. Bouché, H.-U. Reißig*
Synthesis of Novel Carbohydrate Mimetics via 1,2-Oxazines
Pure Appl. Chem. 2012, 84, 23 – 36.
M. Roskamp, S. Enders, F. Pfrengle, S. Yekta. V. Dekaris, J. Dernedde, H.-U. Reißig, S. Schlecht*
Multivalent Interaction and Selectivities in Selectin Binding of Functionalized Gold Colloids Decorated with Carbohydrate Mimetics
Org. Biomol. Chem. 2011, 9, 7448 – 7456.
M. K. Bera, P. Hommes, H.-U. Reißig*
In Search of Oligo(2-thienyl)-Substituted Pyridine Derivatives: A Modular Approach to Di-, Tri- and Tetra(2-thienyl)pyridines
Chem. Eur. J. 2011, 17, 11838 – 11844.
C. Eidamshaus, R. Kumar, M. K. Bera, H.-U. Reißig*
A Practical Two-Step Procedure for the Preparation of Enantiopure Pyridines: Multicomponent Reactions of Alkoxyallenes, Nitriles and Carboxylic Acids followed by a Cyclocondensation Reaction
Beilstein J. Org. Chem. 2011, 7, 962 – 975.
T. Lechel, M. Gerhard, D. Trawny, B. Brusilowskij, L. Schefzig, R. Zimmer, J. P. Rabe, D. Lentz, C. A. Schalley, H.-U. Reißig*
Synthesis of 5-Acetyloxazoles and 1,2-Diketones from β-Alkoxy-β-ketoenamides and Their Subsequent Transformations
Chem.Eur. J. 2011, 17, 7480 – 7491.
V. Dekaris, R. Pulz, A. Al-Harrasi, D. Lentz, H.-U. Reißig*
Stereoselective Synthesis of Aza, Amino and Imion Sugar Derivatives by Hydroboration of 3,6-Dihydro-2H-1,2-oxazines as Key Reaction
Eur. J. Org. Chem. 2011, 3210 – 3219.
A. Al-Harrasi, L. Bouché, R. Zimmer, H.-U. Reißig*
β-Alkoxy-γ-amino Aldehydes by Internal Redox Ring Cleavages of Carbohydrate-Derived Enantiopure 1,2-Oxazines and Preparation of Heterocycles with Aminopolyol Side Chain
Synthesis 2011, 109 – 118.
M. Brasholz, B. Dugovič , H.-U. Reißig*
3-Alkoxy-2,5-dihydrofurans by Gold-Catalyzed Allenyl Cyclizations and Their Transformation into 1,4-Dicarbonyl Compounds, Cyclopentenones, and Butenolides
Synthesis 2010, 3855 – 3864.
F. Pfrengle, H.-U. Reißig*
Internally Protected Amino Sugar Equivalents from Enantiopure 1,2-Oxazines: Synthesis of Variably Configured Carbohydrates with C-Branched Amino Sugar Units
Chem. Eur. J. 2010, 16, 11915 – 11925.
T. Lechel, H.-U. Reißig*
Synthesis of Heterocycles via Alkoxyallenes
Pure Appl. Chem. 2010, 82, 1835 – 1844.
R. Zimmer, T. Lechel, G. Rancan, M. K. Bera, H.-U. Reißig*
Preparation of Pyrimidine-N-oxides by Condensation of Functionalized Enamides with Hydroxylamine Hydrochloride
Synlett 2010, 1793 – 1796.
M. K. Bera, H.-U. Reißig*
A Route to Alkenyl-Substituted 4-Hydroxypyridine and Pyrimidine Derivatives via Three-Component Access to β-Alkoxy-β-ketoenamides
Synthesis 2010, 2129 – 2138.
T. Lechel, J. Dash, C. Eidamshaus, I. Brüdgam, D. Lentz, H.-U. Reißig*
A Three-component Synthesis of β-Alkoxy-β-keto-enamides - Flexible Precoursors for 4-Hydroxypyridine Derivatives and their Palladium-catalysed Reactions
Org. Biomol. Chem. 2010, 8, 3007 – 3014.
T. Lechel, I. Brüdgam, H.-U. Reißig*
Preparation of pyridine-3,4-diols, their crystal packing and their use as precursors for palladium-catalyzed cross-coupling reactions
Beilstein Journal of Organic Chemistry 2010, 6, No. 42.
T. Lechel, H.-U. Reißig*
New 5-Alkoxypyrimidine Derivatives from β-Alkoxy β-Keto Enamides and Ammonium Salts
Eur. J. Org. Chem. 2010, 2555 – 2564.
T. Lechel, J. Dash, P. Hommes, D. Lentz, H.-U. Reißig*
Three-Component Synthesis of Perfluoroalkyl- or Perfluoroaryl-Substituted 4-Hydroxypyridine Derivatives and Their Palladium-Catalyzed Coupling Reactions
J. Org. Chem. 2010, 75, 726 – 732.
F. Pfrengle, H.-U. Reißig*
Amino Sugars and their Mimetics via 1,2-Oxazines
Chem. Soc. Rev., 2010, 39, 549 – 557.
E. Moreno-Clavijo, A. T. Carmona, H.-U. Reißig, A. J. Moreno-Vargas, E. Alvarez, I. Robina*
Allenyl Sulfones and Allenyl Sulfides in the Synthesis of 3-Pyrrolines. A Novel Nucleophilic [3 + 2] Cycloaddition on Allenyl Sulfones Giving Rearranged Cycloadducts
Org. Lett. 2009, 11, 4778 – 4781.
A. Al-Harrasi, S. Fischer, R. Zimmer, H.-U. Reißig*
Ring Enlargement of Carbohydrate-Derived 1,2-Oxazines to Enantiopure 5-Bromo-1,2-oxazepines and Subsequent Palladium-Catalyzed Reactions
Synthesis 2010, 304 – 314.
V. Dekaris, B. Bressel, H.-U. Reißig*
Acid Mediated Transformations of Enantiopure 3,6-Dihydro-2H-1,2-oxazines into Functionalized Aminotetrahydrofuran Derivatives
Synlett 2010, 47 – 50.
V. Dekaris, H.-U. Reißig*
Stereocontrolled Syntheses of Enantiopure Polyhydroxylated Azetidines via 1,2-Oxazines
Synlett 2010, 42 – 46.
A. Al-Harrasi, F. Pfrengle, V. Prisyazhnyuk, S. Yekta, P. Koóš, H.-U. Reißig*
Enantiopure Aminopyrans by a Lewis Acid Promoted Rearrangement of 1,2-Oxazines: Versatile Building Blocks for Oligosaccharide and Sugar Amino Acid Mimetics
Chem. Eur. J. 2009, 15, 11632 – 11642
V. Prisyazhnyuk, M. Jachan, I. Brüdgam, R. Zimmer, H.-U. Reißig*
Addition of Lithiated Methoxyallene to Aziridines – A Novel Access to Enantiopure Piperidine and β-Amino Acid Derivatives
Collect. Czech. Chem. Commun, 2009, 74, 1069 – 1080.
M. Brasholz, H.-U. Reißig*
Alkoxyallene-Based De Novo Synthesis of Rare Deoxy Sugars: New Routes to L-Cymarose, L-Sarmentose, L-Diginose and L-Oleandrose
Eur. J. Org. Chem. 2009, 3595– 3604.
T. Lechel, D. Lentz, H.-U. Reißig*
Three-Component Synthesis of Highly Functionalized 5-Acetyloxazoles
Chem. Eur. J. 2009, 15, 5432 – 5435.
C. Eidamshaus, H.-U. Reißig*
Hihgly Funtionalized Enantiopure 4-Hydroxypyridine Derivatives by a Versatile Three-Component Synthesis
Adv. Synth. Catal. 2009, 351, 1162 - 1166.
F. Pfrengle, D. Lentz, H.-U. Reißig*
Stereodivergente De-novo-Synthese verzweigter Aminozucker durch Lewis-Säure-induzierte Umlagerung von 1,2-Oxazinen
Angew. Chem. 2009, 121, 3211 - 3215.
F. Pfrengle, D. Lentz, H.-U. Reißig*
Stereodivergent De novo Synthesis of Branched Amino Sugars by Lewis Acid promoted Rearrangement of 1,2-Oxazines
Angew. Chem. Int. Ed. 2009, 48, 3165 - 3169.
T. Lechel, S. Möhl, H.-U. Reißig*
A Concise Synthesis of Alkoxy-Substituted Pyrimidine Derivatives Based upon a Three-Component Access to Functionalized Enamides
Synlett 2009, 1059 – 1062.
B. Bressel, H.-U. Reißig*
A New Approach to Neuraminic Acid Analogues via 1,2-Oxazines
Org. Lett. 2009, 11, 527 – 530.
M. Brasholz, H.-U. Reißig,* R. Zimmer
Sugars, Alkaloids and Heteroaromatics: Exploring Heterocyclic Chemistry with Alkoxyallenes
Acc. Chem. Res. 2009, 42, 45 – 56.
F. Pfrengle, A. Al-Harrasi, I. Brüdgam, H.-U. Reißig*
Unusual Enantiopure Heterocyclic Skeletons via Lewis Acid Promoted Rearrangements of 1,3-Dioxolanyl-Substituted 1,2-Oxazines
Eur. J. Org. Chem. 2009, 282 – 291.
F. Pfrengle, V. Dekaris, L. Schefzig, R. Zimmer, H.-U. Reißig*
Indium Trichloride Mediated Cleavage of Acetonides in the Presence of Acid-Labile Functional Groups – Enhancing the Synthetic Utility of 1,3-Dioxolanyl-Substituted 1,2-Oxazines
Synlett 2008, 2965– 2968.
J. Dash, I. Brüdgam, H. Hartl, H.-U. Reißig*
Crystal structure of 1,4-bis[3-methoxy-4(4-methoxyphenyl)-6-(trifluoromethyl)-pyridin-2-yl]benzene, C₃₄H₂₆F₆N₂O₄Z.
Kristallogr. NCS 2008, 223, 347.
R. Zimmer, M. Taszarek. L. Schefzig, H.-U. Reißig*
Reaction of a Polycyclic Diketone with Lithiated Methoxyallene: Synthesis of New Functionalized Cage Compounds
Synlett, 2008, 2046 – 2050.
T. Lechel, J. Dash, I. Brüdgam, H.-U. Reißig*
Novel Furopyridine Derivatives via Sonogashira Reactions of Functionalized Pyridines
Eur. J. Org. Chem. 2008, 3647– 3655.
B. Dugovič, H.-U. Reißig*
A New Alkoxyallene-Based [3+2] Approach to the Synthesis of Highly Substituted Cyclopentenones
Synlett 2008, 769 – 773.
M. Gwiazda, H.-U. Reißig*
Highly Substituted Imidazole Derivatives from a New Four-Component Synthesis Employing Methoxyallene
Synthesis 2008, 990 – 994.
B. Bressel, B. Egart, A. Al-Harrasi, R. Pulz, H.-U. Reißig,* I. Brüdgam
Acid-Induced and Reductive Transformations of Enantiopure 3,6-Dihydro-2H-1,2-oxazines – Synthesis of Dideoxyamino Carbohydrate Derivatives
Eur. J. Org. Chem. 2008, 467 – 474.
B. Dugovič, L. Fišera, H.-U. Reißig*
1,3-Dipolar Cycloadditions of N-Benzyl-2,3-O-isopropylidene-D-glyceraldehyde Nitrone to Methoxyallene – Control of Site- and Diastereoselectivity of Isoxazolidine Formation by Lewis Acids
Eur. J. Org. Chem. 2008, 277 – 284.
S. Yekta, V. Prisyazhnyuk, H.-U. Reißig*
Simple Modifications of Enantiopure 1,2-Oxazines Leading to Building Blocks for Carbohydrate and Peptide Mimetics
Synlett 2007, 2069 – 2072.
M. Brasholz, H.-U. Reißig*
Refined Protocols for the Preparation of 3-Alkoxy-2,5-dihydrofurans, Allylic Oxidation to β-Alkoxybutenolides and Short Synthesis of (±)-Annularin H
Synlett 2007, 1294 - 1298.
M. Brasholz, H.-U. Reißig*
Oxidative Spaltung von 3-Alkoxy-2,5-dihydrofuranen und ihre Anwendung in der
De-novo-Synthese seltener Monosaccharide am Beispiel von L-Cymarose
Angew. Chem. 2007, 119, 1659 – 1662; Angew. Chem. Int. Ed. 2007, 46, 1634 - 1637.
F. Pfrengle, A. Al-Harrasi, H.-U. Reißig*
Lewis Acid Promoted Rearrangements of 1,3-Dioxolanyl-Substituted 1,2-Oxazines
into Novel Products with 1,3,6-Trioxa-7-azacyclopenta[cd]indene Skeletons
Synlett 2006, 3498 – 3500.
S. Sörgel, C. Azap, H.-U. Reißig*
Synthesis of Bisbenzannulated Spiroketals - Model Studies for a Modular Approach
to Rubromycins
Org. Lett. 2006, 8, 4875 - 4878.
S. Kaden, H.-U. Reißig*
Efficient Approach to the Azaspirane Core of FR 901483
Org. Lett. 2006, 8, 4763 - 4766.
S. Sörgel, C. Azap, H.-U. Reißig*
Preparation of Highly Alkoxy-Substituted Naphthaldehyde Derivatives - A
Regioselective Approach to Building Blocks for the Synthesis of Rubromycins
Eur. J. Org. Chem. 2006, 4405 - 4418.
M. A. Chowdhury, H.-U. Reißig*
Syntheses of Highly Substituted Furan and Pyrrole Derivatives via
Lithiated 3-Aryl-1-methoxyallenes: Application to the Synthesis of Codonopsinine
Synlett 2006, 2383 - 2386.
M. Gwiazda, H.-U. Reißig*
A Four-Component Synthesis of Highly Substituted Imidazole Derivatives
Synlett 2006, 1683 - 1686.
M. A. Chowdhury, I. Brüdgam, H. Hartl, H.-U. Reißig*
Crystal structure of (3R,6S,4'S-2-benzyl-3-(2',2'-dimethyl[1',3']dioxolan-
4'-yl)-4-methoxy-6-phenyl-3,6- dihydro-2H-1,2-oxazine, C₂₃H₂₇NO₄
Z. Kristallogr. NCS 2006, 221, 213 - 214.
A. Al-Harrasi, I. Brüdgam, H. Hartl, H.-U. Reißig*
Crystal structure of 3S,4S,5R,6S,7R-5-amino-6-(tert-butyldimetylsiloxy)-
7(tert-butyldimetyl-siloxymethyl)-3-hydroxymethyl-2,2-dimethyloxepan-
4-ol, C₂₂H₄₉NO₅Si₂
Z. Kristallogr. NCS 2006, 221, 131 - 132.
S. Kaden, H.-U. Reißig*, I. Brüdgam, H. Hartl
Additions of Lithiated Alkoxyallenes to Phthalimide: A New Synthesis of
Pyrroloisoindolones and an Unusual Olefination Reaction
Synthesis 2006, 1351 - 1359.
A. Al-Harrasi, I. Brüdgam, H. Hartl, H.-U. Reißig*
Crystal Structure of 3S,4'S,6'S-2-benzyl-3-[(tert-butyldimetylsiloxy)- 2',2'-dimethyl-1,3-dioxolan-4'-yl)-6'-methyl]-4[2-[(trimethylsilyl)ethoxy]- 3,6-dihydro-2H-1,2-oxazine, C₂₈H₄₉NO₅Si₂
Z. Kristallogr. NCS 2006, 221, 12 - 14.
Patent:
O. Flögel, H.-U. Reißig
Substituierte Pyridine
Deutsches Patentamt (DE 10336497 vom 03.03.2005).
R. Zimmer*, H.-U. Reißig
1-Methoxyallenyllithium
in: Electronic Encyclopedia of Reagents for Organic Synthesis
John Wiley & Sons, Chichester, 2005.
A. Al-Harrasi, I. Brüdgam, H. Hartl, H.-U. Reißig*
Crystal structure of 1R,5S,8R,9S-8-azidomethyl-2-benzyl-6,6-dimethyl-3,7-dioxa-
2-azabicyclo[3.3.1]nonan-9-ol, C₁₆H₂₂N₄O₃
Z. Kristallogr. NCS 2005, 220, 599 – 600.
A. Al-Harrasi, H.-U. Reißig*
Enantiomerenreine Kohlenhydratmimetika durch Lewis-Säure-induzierte Umlagerung von 1,3-dioxolanylsubstitutierten 1,2-Oxazinen
Angew. Chem. 2005, 117, 6383 – 6387.
A. Al-Harrasi, H.-U. Reißig*
Ring Enlargement of 1,2-Oxazines to Enantiopure 1,2-Oxazepine Derivatives
and their Palladium-Catalyzed Couplings
Synlett 2005, 2376 - 2378.
S. Kaden, M. Brockmann, H.-U. Reißig*
Synthesis of Enantiopure 2-Substituted Pyrrolidin-3-ones via Lithiated
Alkoxyallenes - An Auxilary Based Synthesis of Both Enantiomers of the Antibiotic Anisomycin.
Helv. Chim. Acta 2005, 88, 1826 - 1838.
A. Al-Harrasi, H.-U. Reißig*
Synthesis of Enantiopure Functionalized β-Alkoxy γ -Amino Aldehydes by a New Internal Redox Ring Cleavage of Carbohydrate Derived 1,2-Oxazines
Synlett 2005, 1152 - 1154.
M. Helms, W. Schade, R. Pulz, T. Watanabe, A. Al-Harrasi, L. Fisera,
I. Hlobilová, G. Zahn, H.-U. Reißig*
Stereodivergent Syntheses of Highly Substituted Enantiopure
4-Alkoxy-3,6-dihydro-2H-1,2-oxazines by Addition of Lithiated Alkoxyallenes to Carbohydrate-Derived Aldonitrones
Eur. J. Org. Chem. 2005, 1003 - 1019.
M. Helms, H.-U. Reißig*
Ozonolyses of Enantiopure 4-Alkoxy-3,6-dihydro-2H-1,2-oxazines: An Expedient Route to Functionalized-Amino-β-hydroxy Esters
Eur. J. Org. Chem. 2005, 998-1001.
C. Azap, P. Luger*, H.-U. Reißig, A. Wagner
Crystal Structure of 4,7,8-Trimethoxy-3-hydroxyspiro[1-benzofuran-2,2'-
chromane] chloroform disolvate, C₁₉H₂₀O₆ · 2 CHCl₃
Z. Kristallogr. NCS 2004, 219, 495 - 496.
C. Azap, P. Luger*, H.-U. Reißig, A. Wagner
Crystal Structure of 4,7-Dimethoxy-3-hydroxyspiro[1-benzofuran-2,2'-chromane] chloroform solvate
(1 : 1/3), C₁₈H₁₈O₅ · 1/3 CHCl₃
Z. Kristallogr. NCS 2004, 219, 492 - 494.
R. Zimmer, H.-U. Reißig
Donor-Substituted Allenes
in "Modern Allene Chemistry" (N. Krause, A. S. K. Hashmi, Eds.), S. 425 – 492, WILEY-VCH, Weinheim 2004.
O. Flögel, J. Dash, I. Brüdgam, H. Hartl, H.-U. Reißig*
A New Color of the Synthetic Chameleon Methoxyallene: Synthesis of Trifluoromethyl-Substituted Pyridinol Derivatives - An Unusual Reaction Mechanism, a Remarkable Crystal Packing, and First Palladium-Catalyzed Coupling Reactions
Chem. Eur. J. 2004, 10, 4283 - 4290.
O. Flögel, H.-U. Reißig*
Direct Synthesis of Functionalized Pyrrole Derivatives from Aldehydes, Bis(trimethylsilyl)amide and Methoxyallene
Synlett 2004, 895 - 897.
O. Flögel, H.-U. Reißig*
Preparation of α,β-Unsaturated γ-Keto Aldehydes and New Tetronic Acid and Pyridazine Derivatives by Oxidative Transformations of Alkoxyallene-Based Dihydrofurans
Eur. J. Org. Chem. 2004, 2797 - 2804.
O. Flögel, M. G. Okala Amombo, H.-U. Reißig*, G. Zahn, I. Brüdgam, H. Hartl
A Stereoselective and Short Total Synthesis of the Polyhydroxylated
γ-Amino Acid (–)-Detoxinine Based on Stereoselective Preparation of Dihydropyrrole Derivatives from Lithiated Alkoxyallenes
Chem. Eur. J. 2003, 9, 1405 - 1415.
R. Pulz, S. Cicchi, A. Brandi, H.-U. Reißig*
Synthesis of New Enantiopure Bicyclic 1,2-Oxazines by Addition of Lithiated Methoxyallene to Chiral Cyclic Nitrones
Eur. J. Org. Chem. 2003, 1153 - 1156.
R. Pulz, W. Schade, H.-U. Reißig*
Synthesis of Enantiopure Amino Polyols and Pyrrolidine Derivatives from 5-Bromo-1,2-oxazin-4-ones
Synlett 2003, 405 - 407.
R. Pulz, A. Al-Harrasi, H.-U. Reißig*
New Polyhydroxylated Pyrrolidines Derived from Enantiopure 3,6-
Dihydro-2H-1,2-oxazines
Org. Lett. 2002, 4, 2353 - 2355.
R. Pulz, A. Al-Harrasi, H.-U. Reißig*
Acid Promoted Syntheses of New Enatiopure Amino Sugar Derivatives from 3,6-Dihydro-2H-1,2-oxazines
Synlett 2002, 817 - 819.
H.-U. Reißig*, W. Schade, M. G. Okala Amombo, R. Pulz, A. Hausherr
Stereoselective Syntheses of Heterocycles via Metallated Alkoxyallenes
Pure Appl. Chem. 2002, 74, 175 - 180.
A. Hausherr, B. Orschel, S. Scherer, H.-U. Reißig*
Synthesis of Enantiopure 1-Alkoxyallenes and their 3-Alkylated Derivatives
Synthesis 2001, 1377 - 1385.
R. Pulz, T. Watanabe, W. Schade, H.-U. Reißig*
A Stereodivergent Synthesis of Enantiopure 3-Methoxypyrrolidines and
3-Methoxy-2,5-dihydropyrroles from 3,6-Dihydro-2H-1,2-oxazines
Synlett 2000, 983 - 986.
H.-U. Reißig*, S. Hormuth, W. Schade, M. Okala Amombo, T. Watanabe, R. Pulz, A. Hausherr,
R. Zimmer
Stereoselective Syntheses of Heterocycles with Lithiated Methoxyallene
Lectures in Heterocyclic Chemistry Vol XVI in J. Heterocycl. Chem. 2000, 37, 597 - 606.
H.-U. Reißig
Lithiiertes Methoxyallen - ein unglaublich vielseitiger Baustein
GIT Labor-Fachzeitschrift 2000, 44, 254 - 256.
R. Pulz, W. Schade, H.-U. Reißig, O. Rademacher*
Crystal Structure of (3R, 5R, 4'S)-2-Benzyl-5-bromo-3-(2',2'-dimethyl-
1',3'-dioxolan-4'-yl)3,4,5,6-tetrahydro-2H-1,2-oxazin-4-one, C₁₆H₂₀BrNO₄
Z. Kristallogr. NCS 2000, 215, 73 - 74.
M. Okala Amombo, A. Hausherr, H.-U. Reißig*
An Expedient Synthesis of Pyrrole Derivatives by Reaction of Lithiated Methoxyallenes with Imines
Synlett 1999, 1871 - 1874.
W. Schade, H.-U. Reißig*
Stereocontrolled Synthesis of the Taxol C-13 Side Chain: Methyl- (2R,3S)-
3-Benzoylamino-2-hydroxy-3-phenylpropanoate
J. Prakt. Chem. 1999, 341, 685 - 686.
W. Schade, H.-U. Reißig*
A New Diastereoselective Synthesis of Enantiomerically Pure 1,2-Oxazine Derivatives by Addition of Lithiated Methoxyallene to Chiral Nitrones
Synlett 1999, 632 - 634.
W. Schade, H.-U. Reißig, G. Zahn*
Crystal Structure of (5S,9S,13S,14S,1'S)-14-[1-(N,N-Dibenzylamino)ethyl]-
1,8,12,15-tetraoxatrispiro[4.3.3.4]heptadecan-4-one, C₂₉H₃₅NO₅
Z. Kristallogr. 1997, 212, 73 - 74.
S. Hormuth, W. Schade, H.-U. Reißig*
First Synthesis of Enantiomerically Pure Primary Helical Spirocycles Based on the Repetitive Addition of Lithiated Methoxyallene to Chiral 3(2H)-Dihydrofuranone Derivatives
Liebigs Ann. 1996, 2001 - 2006.
S. Hormuth, H.-U. Reißig*, D. Dorsch
Stereoselective Synthesis of (2R,3S)-Norstatine Derivatives by Addition of Lithiated Methoxyallene to Amino Aldehydes and Subsequent Ozonolysis
Liebigs Ann. Chem. 1994, 121 - 127.
S. Hormuth, H.-U. Reißig*
Stereoselective Synthesis of 3(2H)-Dihydrofuranones by Addition of Lithiated Methoxyallene to Chiral Aldehydes
J. Org. Chem. 1994, 59, 67 - 73.
S. Hormuth, H.-U. Reißig, S. Foro, H. J. Lindner*
Crystal Structure of (2S,1'S)-2-[1-(N,N-Dibenzylamino)ethyl]-3(2H)-4,5-
dihydrofuranone, OCH₂CH₂COCHCH(CH₃)NCH₂(C₆H₅)CH₂(C₆H₅)
Z. Kristallogr. 1993, 208, 157 - 160.
S. Hormuth, H.-U. Reißig, S. Foro, H. J. Lindner*
Crystal Structure of (5R,1'S)-5-[1-(N,N-Dibenzylamino)ethyl]-2(3H)-4,5-
dihydrofuranone, CH(CH₂)₂COOCHCH₃NCH₂(C₆H₅)CH₂(C₆H₅)
Z. Kristallogr. 1993, 208, 154 - 156.
S. Hormuth, H.-U. Reißig*, D. Dorsch*
Titaniertes Methoxyallen als neuartiges Homoaldoläquivalent in diastereoselektiven Additionen an chirale Aminoaldehyde
Angew. Chem. 1993, 105, 1513 - 1514.
S. Hormuth, H.-U. Reißig*, D. Dorsch*
Titanated Methoxyallene as Novel Homoaldol Equivalent for Diastereoselective Additions to Chiral Amino Aldehydes
Angew. Chem. Int. Ed. Engl. 1993, 32, 1449 – 1450.
S. Hormuth, H.-U. Reißig*
Diastereoselective Additions of Lithiated Methoxyallene towards Chiral Aldehydes
Synlett 1991, 179 - 180.

Synthesis of Natural Products and Analogues

Publications

•	D. Gladow, S. Senf, J. Wiecko, D. Lentz, R. Zimmer, H.-U. Reißig* New Trifluoromethyl-Substituted Heterocycles by Multicomponent Reactions of Siloxycyclopropanes Chem. Heterocycl. Compd. 2017, 53, 416 – 421.
•	M. Wilsdorf, S. Sörgel, H.-U. Reißig Lessons Learned During Spiroketalization Experiments – Progress and Setbacks in the Preparation of Oxygenated Rubromycins and Synthesis of 3´-Desoxyheliquino-mycinone Eur. J. Org. Chem. 2016, 5757 – 5769.
•	M. Wilsdorf, H.-U. Reißig Towards γ-Rubromycin: Model Studies, Development of a New C₃ Building Block and Synthesis of 4´-Silyl-γ-rubromycin Eur. J. Org. Chem. 2016, 5747 – 5756.
•	M. Wilsdorf, H.-U. Reißig* Model Studies towards New Functionalized Bisbenzannulated [5,6]-Spiroketals Eur. J. Org. Chem. 2016, 1555–1561.
•	M. Jasiński, G. Utecht, A. Fruziński, H.-U. Reißig Three-Step Synthesis of 3-Aminoseptanoside Derivatives Using Lithiated Methoxyallene and δ-Siloxynitrones* Synthesis 2016, 48, 893 – 905.
•	H. R. A. Golf, A. M. Oltmanns, D. H. Trieu, H.-U. Reissig,* A. Wiehe* Synthesis of Functionalized BODIPYs, BODIPY-Corrole, and BODIPY-Porphyrin Arrays with 1,2,3-Triazole Linkers Using the 4-Azido(tetrafluorophenyl)-BODIPY Building Block Eur. J. Org. Chem. 2015, 4224 – 4237.
•	C. Beemelmanns, H.-U. Reissig* Strychnine as Target, Samarium Diiodide as Tool: A Personal Story Chem. Rec. 2015, 15, 872 – 885.
•	H. R. A. Golf, H.-U. Reissig, A. Wiehe Synthesis of SF₅-Substituted Tetrapyrroles, Metalloporphyrins, BODIPYs, and Their Dipyrrane Precursors J. Org. Chem. 2015, 80, 5133 – 5143.
•	C. Beemelmanns, H.-U. Reissig* Evolution of a Short Route to Strychnine by Using the Samarium-Diiodide-Induced Cascade Cyclization as a Key Step Chem. Eur. J. 2015, 21, 8416 – 8425.
•	H. R. A. Golf, H.-U. Reißig, A. Wiehe Nucleophilic Substitution on (Pentafluorophenyl)dipyrromethane: A New Route to Building Blocks for Functionalized BODIPYs and Tetrapyrroles Org. Lett. 2015, 17, 982 – 985.
•	H. R. A. Golf, H.-U. Reißig, A. Wiehe* *Regioselective Nucleophilic Aromatic Substitution Reaction of meso-Pentafluorophenyl-Substituted Porphyrinoids with Alcohols* Eur. J. Org. Chem. 2015, 1548 – 1568.
•	C. N. Rao, D. Lentz, H.-U. Reißig* Synthese polycyclischer tertiärer Carbinamine durch Samariumdiiodid-vermittelte Cyclisierungen von Indolylsulfinylimien Angew. Chem. 2015, 127, 2788 – 2792. C. N. Rao, D. Lentz, H.-U. Reißig* Synthesis of Polycyclic Tertiary Carbinamines by Samarium Diiodide Mediated Cyclizations of Indolyl Sulfinyl Imines Angew. Chem. Int. Ed. 2015, 54, 2750 – 2753.
•	M. Wilsdorf, H.-U. Reißig* Eine konvergente Totalsynthese des Telomerase-Inhibitors (±)-γ-Rubromycin Angew. Chem. 2014, 126, 4420 – 4424. M. Wilsdorf, H.-U. Reißig* A Convergent Total Synthesis of the Telomerase Inhibitor (±)-γ-Rubromycin Angew. Chem. Int. Ed. 2014, 53, 4332 – 4336.
•	M. Jasiński, E. Moreno-Clavijo, H.-U. Reißig* Synthesis of a Series of Enantiopure Polyhydroxylated Bicyclic N-Heterocycles from an l-Erythrose Derived Nitrone and Alkoxyallenes Eur. J. Org. Chem. 2014, 442 – 454.
•	C. Beemelmanns, S. Gross, H.-U. Reißig* *Towards the Core Structure of Strychnos* Alkaloids Using Samarium Diiodide-Induced Reactions of Indole Derivatives** Chem. Eur. J. 2013,19, 17801 – 17808.
•	V. M. Schmiedel, S. Stefani, H.-U. Reißig* Stereodivergent Synthesis of Jaspine B and its Isomers using a Carbohydrate-derived Alkoxyallene as C₃-building Block Beilstein J. Org. Chem. 2013,9, 2564 – 2569.
•	T. H. Ngo, H. Berndt, M. Wilsdorf, D. Lentz, H.-U. Reißig* Linear and Cyclic Hybrids of Alternating Thiophene–Amino Acid Units: Synthesis and Effects of Chirality on Conformation and Molecular Packing Chem. Eur. J. 2013,19, 15155 – 15165.
•	C. Parmeggiani, F. Cardona, L. Giusti, H.-U. Reißig, A. Goti Stereocomplementary Routes to Hydroxylated Nitrogen Heterocycles: Total Syntheses of Casuarine, Australine, and 7-epi-Australine* Chem. Eur. J. 2013, 19, 10595 – 10604.
•	M. H. Beyzavi, C. Nietzold, H.-U. Reißig, A. Wiehe Synthesis of Functionalized trans-A2B2-Porphyrins Using Donor-Acceptor Cyclopropane-Derived Dipyrromethanes Adv. Synth. Catal. 2013, 355, 1409 – 1422.
•	M. Wilsdorf, D. Leichnitz, H.-U. Reißig* Trifluoromethanesulfonic Acid Catalyzed Friedel-Crafts Alkylations of 1,2,4-Trimethoxybenzene with Aldehydes or Benzylic Alcohols Org. Lett. 2013, 15, 2494 – 2497.
•	M. H. Beyzavi, D. Lentz, H.-U. Reißig, A. Wiehe Synthesis of New Functionalized Calix[n]phyrin Macrocycles with Varied Ring Sizes by Using a Sterically Congested Dipyrromethane Chem. Eur. J. 2013, 19, 6203 – 6208.
•	T. H. Ngo, H. Berndt, D. Lentz, H.-U. Reißig* Linear and Cyclic Amides with a Thiophene Backbone: Ultrasound-Promoted Synthesis and Crystal Structures J. Org. Chem. 2012, 77, 9676 – 9683.
•	M. Wilsdorf, H.-U. Reißig* Einfach und dennoch herausfordernd: Neues zur asymmetrischen Synthese von Spiroketalen Angew. Chem. 2012, 124, 9624 – 9626. M. Wilsdorf, H.-U. Reißig* Simple, but Challenging: Recent Developments in the Asymmetric Synthesis of Spiroketals Angew. Chem. Int. Ed. 2012, 51, 9486 – 9488.
•	M. Jasiński, Dieter Lentz, E. Moreno-Clavijo, H.-U. Reißig* Application of L-Erythrose-Derived Nitrones in the Synthesis of Polyhydroxylated Compounds via 3,6-Dihydro-2H-1,2-oxazine Derivatives Eur. J. Org. Chem. 2012, 3304 – 3316.
•	M. Jasiński, Dieter Lentz, H.-U. Reißig* Carbohydrate-Auxiliary Assisted Preparation of Enantiopure 1,2-Oxazine Derivatives and Aminopolyols Beilstein J. Org. Chem. 2012, 8, 662-674.
•	L. Bouché, H.-U. Reißig* Synthesis of Novel Carbohydrate Mimetics via 1,2-Oxazines Pure Appl. Chem. 2012, 84, 23 – 36.
•	C. Beemelmanns, D. Lentz, H.-U. Reißig* Samarium Diiodide Induced Cyclizations of γ-, δ- and ε-Indolyl Ketones: Reductive Coupling, Intermolecular Trapping, and Subsequent Transformations of Indolines Chem. Eur. J. 2011, 17, 9720 – 9730.
•	V. Dekaris, R. Pulz, A. Al-Harrasi, D. Lentz, H.-U. Reißig* Stereoselective Synthesis of Aza, Amino and Imion Sugar Derivatives by Hydroboration of 3,6-Dihydro-2H-1,2-oxazines as Key Reaction Eur. J. Org. Chem. 2011, 3210 – 3219.
•	C. Beemelmanns, H.-U. Reißig* Samarium diiodide induced ketyl-(het)arene cyclisations towards novel N-heterocycles Chem. Soc. Rev., 2011, 40, 2199 – 2210.
•	H. Özbek, D. Lentz, H.-U. Reißig* New Macrocyclic Peptidomimetics Containing 5-Aminothiophene Subunits Eur. J. Org. Chem. 2010, 6319 – 6322.
•	M. Brasholz, B. Dugovič , H.-U. Reißig* 3-Alkoxy-2,5-dihydrofurans by Gold-Catalyzed Allenyl Cyclizations and Their Transformation into 1,4-Dicarbonyl Compounds, Cyclopentenones, and Butenolides Synthesis 2010, 3855 – 3864.
•	C. Beemelmanns, H.-U. Reißig* Eine kurze formale Strychnin-Totalsynthese mit einer Samariumdiiodid-induzierten Kaskadenreaktion als Schlüsselschritt Angew. Chem. 2010, 122, 8195 – 8199. C. Beemelmanns, H.-U. Reißig* A Short Formal Total Synthesis of Strychnine with a Samarium Diiodide Induced Cascade Reaction as the Key Step Angew. Chem. Int. Ed. 2010, 49, 8021 – 8025.
•	F. Pfrengle, H.-U. Reißig* Internally Protected Amino Sugar Equivalents from Enantiopure 1,2-Oxazines: Synthesis of Variably Configured Carbohydrates with C-Branched Amino Sugar Units Chem. Eur. J. 2010, 16, 11915 – 11925.
•	A. Schwanke, C. Murruzzu, B. Zdrazil. R. Zuhse, M. Natek, M. Höltje, H. C. Korting, H.-U. Reißig, H.-D. Höltje, M. Schäfer-Korting* Antitumor Effects of Guanosine-Analog Phosphonates Identified by Molecular Modelling Int. J. Pharm. 2010, 397, 9 – 18.
•	U. K. Wefelscheid, H.-U. Reißig* Synthesis of New Steroid Analogues by Samarium Diiodide Induced Cyclisations of γ-Naphthyl 1,3-Diones Tetrahedron: Asymmetry 2010, 21, 1601 – 1610.
•	F. Pfrengle, H.-U. Reißig* Addition of Lithiated Enol Ethers to Nitrones and Subsequent Lewis Acid Induced Cyclizations to Enantiopure 3,6-Dihydro-2H-pyrans – an Approach to Carbohydrate Mimetics Beilstein Journal of Organic Chemistry 2010, 6, No. 75.
•	M. Höltje, A. Richartz, B. Zdrazil, A. Schwanke, B. Dugovič, C. Murruzzu, H.-U. Reißig, H. C. Korting, B. Kleuser, H.-D. Höltje, M. Schäfer-Korting* Human Polymerase α-Inhibitors for Skin Tumors. Part 2. Modeling, Synthesis and Influence on Normal and Transformed Keratinocytes of New Thymidine and Purine Derivatives J. Enzym. Inhib. Med. Chem., 2010, 25 (2), 250-265.
•	V. Dekaris, H.-U. Reißig* Stereocontrolled Syntheses of Enantiopure Polyhydroxylated Azetidines via 1,2-Oxazines Synlett 2010, 42 – 46.
•	F. Pfrengle, D. Lentz, H.-U. Reißig* A New Ring Closure Approach to Enantiopure 3,6-Dihydro-2H-pyrans: Stereodivergent Access to Carbohydrate Mimetics Org. Lett. 2009, 11, 5534 – 5537.
•	V. Prisyazhnyuk, M. Jachan, I. Brüdgam, R. Zimmer, H.-U. Reißig* Addition of Lithiated Methoxyallene to Aziridines – A Novel Access to Enantiopure Piperidine and β-Amino Acid Derivatives Collect. Czech. Chem. Commun, 2009, 74, 1069 – 1080.
•	M. Brasholz, H.-U. Reißig* Alkoxyallene-Based De Novo Synthesis of Rare Deoxy Sugars: New Routes to L-Cymarose, L-Sarmentose, L-Diginose and L-Oleandrose Eur. J. Org. Chem. 2009, 3595– 3604.
•	J. Dash, H.-U. Reißig* A New and Flexible Synthesis of 4-Hydroxypyridines: Rapid Access to Caerulomycins A, E and Functionalized Terpyridines Chem. Eur. J. 2009, 15, 6811 – 6814.
•	F. Pfrengle, D. Lentz, H.-U. Reißig* Stereodivergente De-novo-Synthese verzweigter Aminozucker durch Lewis-Säure-induzierte Umlagerung von 1,2-Oxazinen Angew. Chem. 2009, 121, 3211 - 3215.
	F. Pfrengle, D. Lentz, H.-U. Reißig* Stereodivergent De novo Synthesis of Branched Amino Sugars by Lewis Acid promoted Rearrangement of 1,2-Oxazines Angew. Chem. Int. Ed. 2009, 48, 3165 - 3169.
•	V. Blot, U. Jacquemard, H.-U. Reißig,* B. Kleuser Practical Syntheses of Sphingosine-1-Phosphate and Analogues Synthesis 2009, 759 – 766.
•	J. Dernedde, S. Enders, H.-U. Reißig, M. Roskamp, S. Schlecht,* S. Yekta Inhibition of selectin binding by colloidal gold with functionalized shells Chem. Commun. 2009, 932 – 934.
•	B. Bressel, H.-U. Reißig* A New Approach to Neuraminic Acid Analogues via 1,2-Oxazines Org. Lett. 2009, 11, 527 – 530.
•	M. Brasholz, H.-U. Reißig,* R. Zimmer Sugars, Alkaloids and Heteroaromatics: Exploring Heterocyclic Chemistry with Alkoxyallenes Acc. Chem. Res. 2009, 42, 45– 56.
•	C. Venkatesh, H.-U. Reißig* Model Studies for the Synthesis of Heliquinomycin: Preparation of New Spiroketals Synthesis 2008, 3605 – 3614.
•	F. Aulenta, U. K. Wefelsched, I. Brüdgam, H.-U. Reißig* Nitrogen-Containing Tricyclic and Tetracyclic Compounds via Stereoselective Samarium Diiodide Promoted Cyclizations of Quinolyl-Substituted Ketones – A New Access to Azasteroids Eur. J. Org. Chem. 2008, 2325 - 2335.
•	U. K. Wefelscheid, H.-U. Reißig* Pentacyclic Compounds by Samarium Diiodide-Induced Cascade Cyclizations of Naphthyl-Substituted 1,3-Diones Adv. Synth. Catal, 2008, 250, 65 – 69.
•	M. Brasholz, S. Sörgel, C. Azap, H.-U. Reißig* Rubromycins: Structurally Intriguing, Biologically Valuable, Synthetically Challenging Antitumour Antibiotics Eur. J. Org. Chem. 2007, 3801 – 3814.
•	F. Aulenta, M. Berndt, I. Brüdgam, H. Hartl, S. Sörgel, H.-U. Reißig* A New, Efficient and Stereoselective Synthesis of Tricyclic and Tetracyclic Compounds by Samarium Diiodide Induced Cyclisations of Naphthyl-Substituted Arylketones – An Easy Access to Steroid-Like Skeletons Chem. Eur. J. 2007, 13, 6047 – 6062.
•	S. Sörgel, I. Brüdgam, H. Hartl, H.-U. Reißig* Crystal structure of 2-bromo-1,4,5,7,8-pentamethoxynaphthalene, C₁₀H₂Br(OCH₃)₅Z. Kristallogr. NCS 2006, 221, 278 – 280.
•	S. Sörgel, C. Azap, H.-U. Reißig Synthesis of Bisbenzannulated Spiroketals – Model Studies for a Modular Approach to Rubromycins Org. Lett. 2006, 8, 4875 – 4878.
•	S. Kaden, H.-U. Reißig* Efficient Approach to the Azaspirane Core of FR 901483 Org. Lett. 2006, 8, 4763 – 4766.
•	S. Sörgel, C. Azap, H.-U. Reißig* Preparation of Highly Alkoxy-Substituted Naphthaldehyde Derivatives – A Regioselective Approach to Building Blocks for the Synthesis of Rubromycins Eur. J. Org. Chem. 2006, 4405 – 4418.
•	M. A. Chowdhury, H.-U. Reißig* Syntheses of Highly Substituted Furan and Pyrrole Derivatives via Lithiated 3-Aryl-1-methoxyallenes: Application to the Synthesis of Codonopsinine. Synlett 2006, 2383 – 2386.
•	M. Brasholz, X. Luan, H.-U. Reißig Towards the Rubromycins: An Efficient Synthesis of a Suitable Isocoumarin Precursor, its Lactam Analogue, and Palladium-Catalyzed Couplings* Synthesis 2005, 3571 – 3580.
•	S. Kaden, M. Brockmann, H.-U. Reißig* Synthesis of Enantiopure 2-Substituted Pyrrolidin-3-ones via Lithiated Alkoxyallenes – An Auxilary Based Synthesis of Both Enantiomers of the Antibiotic Anisomycin. Helv. Chim. Acta 2005, 88, 1826 – 1838.
•	M. Brasholz, H.-U. Reißig* An Expedient and Short Synthesis of a 6-Iodo Isocoumarin Building Block for the Rubromycin Family and its First Palladium-Catalyzed Couplings Synlett 2004, 2736 – 2738.
•	M. Berndt, I. Hlobilová, H.-U. Reißig* Stereoselective Formation of Tri- and Tetracycles by Samarium Diiodide-Induced Cyclizations of Naphthyl-Substituted Ketones Org. Lett. 2004, 6, 957 – 960. >
•	O. Flögel, M. G. Okala Amombo, H.-U. Reißig, G. Zahn, I. Brüdgam, H. Hartl A Stereoselective and Short Total Synthesis of the Polyhydroxylated γ-Amino Acid (-)-Detoxinine Based on Stereoselective Preparation of Dihydropyrrole Derivatives from Lithiated Alkoxyallenes* Chem. Eur. J. 2003, 9, 1405 – 1415.
•	W. Schade, H.-U. Reißig* Stereocontrolled Synthesis of the Taxol C-13 Side Chain: Methyl (2R,3S)-3-Benzoylamino-2-hydroxy-3-phenylpropanoate J. Prakt. Chem. 1999, 341, 685 – 686.
•	J. Schnaubelt, B. Frey, H.-U. Reißig* Formal Total Synthesis of (+)-Dihydromevinolin via a Chelate-Controlled Intramolecular Diels-Alder Reaction as the Key Step Helv. Chim. Acta 1999, 82, 666 – 676.
•	H. Angert, R. Czerwonka, H.-U. Reißig* Additions of Silyl Enol Ethers to β-Formyl Esters – A Chelate-Controlled Synthesis of the Pheromone (+)-Eldanolide. Liebigs Ann. 1996, 259 – 263.
•	K. Paulini, H.-U. Reißig* Preparation of Novel Lipophilic GABA-Analogues Containing Cyclopropane Rings via Cyclopropanation of N-Silylated Unsaturated Amines J. prakt. Chem. 1995, 337, 55 – 59.
•	K. Paulini, H.-U. Reißig* Synthesis of Dipeptides Containing Novel Cyclopropyl- and Cyclopropenyl-Substituted β- und γ-Amino Acids Liebigs Ann. Chem. 1994, 549 – 554.
•	A. G. Beck-Sickinger, E. Hoffmann, K. Paulini, H.-U. Reißig, K.-D. Willim, H. A. Wieland, G. Jung High-Affinity Analogues of Neuropeptide Y Containing Conformationally Restricted Non-Proteinogenic Amino Acids* Biochem. Soc. Trans. 1994, 22, 145 – 149.
•	J. Schnaubelt, R. Zschiesche, H.-U. Reißig, H. J. Lindner, J. Richter Synthese von Östronderivaten aus Siloxycyclopropancarbonsäureestern* Liebigs Ann. Chem. 1993, 61 – 70.
•	K. Paulini, H.-U. Reißig* Efficient Synthesis of a Novel GABA Analogue Incorporating a Cyclopropene Ring Synlett 1992, 505 – 506.
•	R. Zschiesche, T. Hafner, H.-U. Reißig* Conversion of Polyfunctional Nitroalkanes into Carbonyl Compounds – Synthesis of the Pheromone Chalcogran and of Key Building Blocks for the Macrolides Pyrenophorin and Vermiculine Liebigs Ann. Chem. 1988, 1169 – 1173.
•	R. Zschiesche, H.-U. Reißig* *Eine Synthexe von rac-Norbisabolid* Liebigs Ann. Chem. 1987, 387 - 388.
•	I. Reichelt, H.-U. Reißig* Neue Chrysanthemumsäurederivative druch Deprotonierung-Alkylierung Liebigs Ann. Chem. 1985, 650 - 652.

Synthesis of Novel Pyridine Derivatives

Publications

	J. Klein, A. Stuckmann, S. Sobottka, L. Suntrup, M. van der Meer, P. Hommes, H.-U. Reißig, B. Sarkar* Ruthenium Complexes with Strongly Electron-Donating Terpyridine Ligands: Effect of the Working Electrode on Electrochemical and Spectroelectrochemical Properties Chem. Eur. J. 2017, 23, 12314 – 12325.
	S. Aroua, T. K. Todorova, V. Mougel, P. Hommes, H.-U. Reißig, M. Fontecave* New Cobalt-Bisterpyridyl Catalysts for Hydrogen Evolution Reaction ChemCatChem 2017, 9, 2099 – 2105.
	S. Aroua, T. K. Todorova, P. Hommes, L.-M. Chamoreau, H.-U. Reißig, V. Mougel, M. Fontecave* Synthesis, Characterisation and DFT Analysis of Bisterpyridyl-Based Molecular Cobalt Complexes Inorganic Chem. 2017, 56, 5930 – 5940.
	T. Pecchioli, F. Cardona, H.-U. Reißig, R. Zimmer, A. Goti Alkoxyallene-Based Stereodivergent Syntheses of (–)-Hyacinthacine B₄ and of Putative Hyacinthacine C₅ Epimers – Proposal of Hyacinthacine C₅ Structure J. Org. Chem. 2017, 82, 5835 – 5844.
•	S. Aroua, T. K. Todorova, P. Hommes, L.-M. Chamoreau, H.-U. Reißig, V. Mougel, M. Fontecave* Synthesis, Characterisation and DFT Analysis of Bisterpyridyl-Based Molecular Cobalt Complexes Inorganic Chem. 2017, 56, 5930 – 5940.
•	T. Pecchioli, F. Cardona, H.-U. Reißig, R. Zimmer, A. Goti Alkoxyallene-Based Stereodivergent Syntheses of (–)-Hyacinthacine B₄ and of Putative Hyacinthacine C₅ Epimers – Proposal of Hyacinthacine C₅ Structure J. Org. Chem. 2017, 82, 5835 – 5844.
•	H.-U. Reißig, M. Domínguez* N-Methylpyridinium-4-phenolates: Generation of a Betaine Dye Library Bearing Different Spacer Units and Their Solvatochromism ChemistrySelect 2016, 1, 5270 – 5275.
•	P. Hommes, H.-U. Reißig* Synthesis of Highly Functionalized 2,2´-Bipyridines by Cyclocondensation of β-Ketoenamides – Scope and Limitations Beilstein J. Org. Chem. 2016, 12, 1170 – 1177.
•	P. Hommes, H.-U. Reißig* Functionalization of Highly Substituted 2,2´:6,6´,2´´-Terpyridine Derivatives Eur. J. Org. Chem. 2016, 338 – 342.
•	G. Podolan, L. Hettmanczyk, P. Hommes, B. Sarkar,* H.-U. Reißig* Synthesis and (Spectro)electrochemistry of New Ferrocenyl-Substituted Pyridine Derivatives Eur. J. Org. Chem. 2015, 7317 – 7323.
•	D. Trawny, M. Quennet, N. Rades, D. Lentz, B. Paulus, H.-U. Reissig* Syntheses, Structures and Conformational Dynamics of 1,3,5-Tris(3‘‘-ethynylbi-phenyl-2‘-yl)benzene Derivatives Eur. J. Org. Chem. 2015, 4667 – 4674.
•	M. Gensler, C. Eidamshaus, M. Taszarek, H.-U. Reissig, J. P. Rabe* Mechanical Stability of Bivalent Transition Metal Complexes Analyzed by Single-Molecule Force Spectroscopy Beilstein J. Org. Chem. 2015, 11, 817 – 827.
•	J. Dash, D. Trawny, J. P. Rabe, H.-U. Reissig* C₃-Symmetric Pyridine and Bipyridine Derivatives: Simple Preparation by Cyclocondensation and 2D Self-Assembly at a Solution-Graphite Interface Synlett 2015, 26, 1486 – 1489.
•	M. Gensler, C. Eidamshaus, A. Galstyan, E.-W. Knapp, H.-U. Reißig, J. P. Rabe Mechanical Rupture of Mono- and Bivalent Transition Metal Complexes in Experiment and Theory J. Phys. Chem. C 2015, 119, 4333 – 4343.
•	D. Trawny, P. Schlexer, K. Steenbergen, J. P. Rabe, B. Paulus, H.-U. Reißig* Dense or Porous Packing? Two-Dimensional Self-Assembly of Star-Shaped Mono-, Bi-, and Terpyridine Derivatives ChemPhysChem 2015, 16, 949 – 953.
•	D. Trawny, V. Kunz, H.-U. Reißig* Modular Syntheses of Star-Shaped Pyridine, Bipyridine, and Terpyridine Derivatives by Employing Sonogashira Reactions Eur. J. Org. Chem. 2014, 6295 – 6302.
•	D. Trawny, L. Vandromme, J. P. Rabe,* H.-U. Reissig* The Side Chain Makes the Difference: Investigation of the 2D Self-Assembly of 1,3,5-Tris[4-(4-pyridinyl)phenyl]benzene Derivatives by Scanning Tunneling Microscopy Eur. J. Org. Chem. 2014, 4985 – 4992.
•	D. Gladow, S. Doniz-Kettenmann, H.-U. Reißig* 1,3-Dipolar Cycloadditions of Ethyl 2-Diazo-3,3,3-trifluoropropanoate to Alkynes and [1,5] Sigmatropic Rearrangements of the Resulting 3H-Pyrazoles: Synthesis of Mono-, Bis- and Tris(trifluoromethyl)-Substituted Pyrazoles Helv. Chim. Acta, 2014, 97, 808 – 821.
•	D. Gladow, H.-U. Reißig* Perfluoroalkyl-Substituted Thiophenes and Pyrroles from Donor-Acceptor Cyclopropanes and Heterocumulenes: Synthesis and Exploration of their Reactivity J. Org. Chem. 2014, 79, 4492 – 4502.
•	L. Bouché, H.-U. Reißig* Synthesis of Di- and Trivalent Carbohydrate Mimetics with Oxepane Substructure by Employing Copper-Catalyzed [3+2] Cycloadditions of Alkynes with Azidooxepanes Eur. J. Org. Chem. *2014,* 3697 – 3703.
•	M. Domínguez, H.-U. Reißig* New 4-Pyridyl Nonaflates as Precursors for Push-Pull Solvatochromik Dyes Synthesis 2014, 46, 1110 – 1106.
•	M. K. Bera, M. Domínguez, P. Hommes, H.-U. Reißig* The Flögel-Three-Component Reaction with Dicarboxylic Acids - An Approach to Bis(β-alkoxy-β - ketoenamides) for the Synthesis of Complex Pyridine and Pyrimidine Derivatives Beilstein J. Org. Chem. 2014, 10, 394 – 404.
•	M. K. Bera, S. L. Gholap, P. Hommes, K. Neuthe, D. Trawny, J. P. Rabe, D. Lentz, R. Zimmer, H.-U. Reißig* Synthesis and Properties of Branched Oligo(2-thienyl)- and Oligo(2,2’-bithien-5-yl)-Substituted Pyridine Derivatives Adv. Synth. Catal. 2013, 355, 3463 – 3474
•	P. Hommes, S. Berlin, H.-U. Reißig* Trimethylsilyl Trifluoromethanesulfonate-Promoted Cyclocondensation of b-Keto-enamides and Subsequent Nonaflation to Pyrid-2-yl and Pyrid-4-yl Nonaflates as Flexible Precursors for Polysubstituted Pyridines Synthesis 2013, 45, 3288 – 3294.
•	S. L. Gholap, P. Hommes, K. Neuthe, H.-U. Reißig* Per(2-thienyl)pyridines: Synthesis and Properties Org. Lett. 2013, 15, 318 – 321.
•	T. Lechel, G. Podolan, B. Brusilowskij, C. A. Schalley, H.-U. Reißig* Unexpected One-Step Formation of Iodo[1,3]dioxolo[4,5-c]pyridine Derivatives by a Hofmann-Löffler-Freytag Reaction: Studies on the Synthesis of a Pyridine-Containing Macrocycle Eur. J. Org. Chem. 2012, 5685 – 5692 .
•	C. Eidamshaus, P. Hommes, H.-U. Reißig* Palladium-Catalyzed Coupling of Pyrid-4-yl Nonaflates with Methyl Diazoacetate Synlett 2012, 1670 – 1674.
•	C. Eidamshaus, T. Triemer, H.-U. Reißig* *Synthesis of 4-Quinolones via Cyclocondensation of Substituted ortho-Amidoacetophenones: A Refit to the Camps Cyclization by Applying Trimethylsilyl Trifluoromethanesulfonate/Triethylamine* Synthesis 2011, 3261 – 3266.
•	I. Linder, M. Gerhard, L. Schefzig, M. Andrä, C. Bentz, H.-U. Reißig,* R. Zimmer A Modular Synthesis of Functionalized Pyridines through Lewis-Acid-Mediated and Microwave-Assisted Cycloadditions between Azapyrylium Intermediates and Alkynes Eur. J. Org. Chem. 2011, 6070 – 6078.
•	C. Eidamshaus, H.-U. Reißig* A Chiral Pool Strategy for the Synthesis of Enantiopure Hydroxymethyl-Substituted Pyridine Derivatives Eur. J. Org. Chem. 2011, 6056 – 6069
•	M. K. Bera, P. Hommes, H.-U. Reißig* In Search of Oligo(2-thienyl)-Substituted Pyridine Derivatives: A Modular Approach to Di-, Tri- and Tetra(2-thienyl)pyridines Chem. Eur. J. 2011, 17, 11838 – 11844.
•	P. Hommes, P. Jungk, H.-U. Reißig* Four-Component Synthesis of Functionalized 2,2’-Bipyridines Based on the Blaise Reaction Synlett 2011, 2311 – 2314.
•	C. Eidamshaus, R. Kumar, M. K. Bera, H.-U. Reißig* A Practical Two-Step Procedure for the Preparation of Enantiopure Pyridines: Multicomponent Reactions of Alkoxyallenes, Nitriles and Carboxylic Acids followed by a Cyclocondensation Reaction Beilstein J. Org. Chem. 2011, 7, 962 – 975.
•	T. Lechel, M. Gerhard, D. Trawny, Boris Brusilowskij, L. Schefzig, R. Zimmer, J. P. Rabe, D. Lentz, C. A. Schalley, H.-U. Reißig* Synthesis of 5-Acetyloxazoles and 1,2-Diketones from β-Alkoxy-β-ketoenamides and Their Subsequent Transformations Chem. Eur. J. 2011, 7480 – 7491.
•	D. Mollenhauer, J. Floß, H.-U. Reißig, E. Voloshina, B. Paulus* Accurate Quantum-Chemical Description of Gold Complexes with Pyridine and its Derivatives J. Comput. Chem. 2011, 32, 1839 – 1845.
•	T. Lechel, H.-U. Reißig* Synthesis of Heterocycles via Alkoxyallenes Pure Appl. Chem. 2010, 82, 1835 – 1844.
•	M. K. Bera, H.-U. Reißig* A Route to Alkenyl-Substituted 4-Hydroxypyridine and Pyrimidine Derivatives via Three-Component Access to β-Alkoxy-β-ketoenamides Synthesis 2010, 2129 – 2138.
•	T. Lechel, J. Dash, C. Eidamshaus, I. Brüdgam, D. Lentz, H.-U. Reißig* A Three-component Synthesis of β-Alkoxy-β-keto-enamides - Flexible Precoursors for 4-Hydroxypyridine Derivatives and their Palladium-catalysed Reactions Org. Biomol. Chem. 2010, 8, 3007 – 3014.
•	T. Lechel, I. Brüdgam, H.-U. Reißig* Preparation of pyridine-3,4-diols, their crystal packing and their use as precursors for palladium-catalyzed cross-coupling reactions Beilstein Journal of Organic Chemistry 2010, 6, No. 42.
•	T. Lechel, J. Dash, P. Hommes, D. Lentz, H.-U. Reißig* Three-Component Synthesis of Perfluoroalkyl- or Perfluoroaryl-Substituted 4-Hydroxypyridine Derivatives and Their Palladium-Catalyzed Coupling Reactions J. Org. Chem. 2010, 75, 726 – 732.
•	T. Lechel, H.-U. Reißig* New 5-Alkoxypyrimidine Derivatives from β-Alkoxy β-Keto Enamides and Ammonium Salts Eur. J. Org. Chem. 2010, 2555 – 2564.
•	R. Zimmer, E. Schmidt, M. Andrä, M.-A. Duhs, I. Linder, H.-U. Reißig* Palladium-catalyzed cross coupling reactions of 4-bromo-6H-1,2-oxazines Beilstein Journal of Organic Chemistry 2009, 5, No. 44.
•	J. Dash, H.-U. Reißig* A New and Flexible Synthesis of 4-Hydroxypyridines: Rapid Access to Caerulomycins A, E and Functionalized Terpyridines Chem. Eur. J. 2009, 15, 6811 – 6814.
•	C. Eidamshaus, H.-U. Reißig* Hihgly Funtionalized Enantiopure 4-Hydroxypyridine Derivatives by a Versatile Three-Component Synthesis Adv. Synth. Catal. 2009, 351, 1162 - 1166.
•	T. Lechel, S. Möhl, H.-U. Reißig* A Concise Synthesis of Alkoxy-Substituted Pyrimidine Derivatives Based upon a Three-Component Access to Functionalized Enamides Synlett 2009, 1059 – 1062.
•	J. Dash, I. Brüdgam, H. Hartl, H.-U. Reißig* Crystal structure of 1,4-bis[3-methoxy-4(4-methoxyphenyl)-6-(trifluoromethyl)-pyridin-2-yl]benzene, C₃₄H₂₆F₆N₂O₄Z. Kristallogr. NCS 2008, 223, 347.
•	T. Lechel, J. Dash, I. Brüdgam, H.-U. Reißig* Novel Furopyridine Derivatives via Sonogashira Reactions of Functionalized Pyridines Eur. J. Org. Chem. 2008, 3647– 3655.
•	L. Vandromme, H.-U. Reißig, S. Gröper, J. P. Rabe Practical Routes to New 2,6-Disubstituted Pyridine Derivatives* Eur. J. Org. Chem. 2008, 2049 - 2055.
•	J. Dash, T. Lechel, H.-U. Reißig* Scope of a Novel Three-Component Synthesis of Highly Functionalized Pyridines Org. Lett. 2007, 9, 5541 – 5544.
•	Patent: O. Flögel, H.-U. Reißig Substituierte Pyridine Deutsches Patentamt (DE 10336497 vom 03.03.2005)
•	O. Flögel, J. Dash, I. Brüdgam, H. Hartl, H. U. Reißig* A New Color of the Synthetic Chameleon Methoxyallene: Synthesis of Trifluoromethyl-Substituted Pyridinol Derivatives – An Unusual Reaction Mechanism, a Remarkable Crystal Packing, and First Palladium-Catalyzed Coupling Reactions Chem. Eur. J. 2004, 10, 4283 – 4290.

Samarium Diiodide Induced Cyclization Reactions

Publications

•	A. J. Achazi, D. Andrae, H.-U. Reißig, B. Paulus A Computational Study of Samarium Diiodide-Induced Cyclizatons of N-Oxoalkyl-Substituted Methyl Indole-3-Carboxylates - A Rationale of the* Diastereoselectivity J. Comput. Chem. 2017, 38, 2693 – 2700.
•	C. N. Rao, C. Bentz, H.-U. Reissig* Lithium Bromide/Water as Additives in Dearomatizing Samarium-Ketyl (Hetero)Arene Cyclizations Chem. Eur. J. 2015, 21, 15951 – 15954.
•	C. Beemelmanns, H.-U. Reissig* Strychnine as Target, Samarium Diiodide as Tool: A Personal Story Chem. Rec. 2015, 15, 872 – 885.
•	C. Beemelmanns, H.-U. Reißig* Evolution of a Short Route to Strychnine by Using the Samarium-Diiodide-Induced Cascade Cyclization as a Key Step Chem. Eur. J. 2015, 21, 8416 – 8425.
•	C. N. Rao, D. Lentz, H.-U. Reißig* Synthese polycyclischer tertiärer Carbinamine durch Samariumdiiodid-vermittelte Cyclisierungen von Indolylsulfinylimien Angew. Chem. 2015, 127, 2788 – 2792. C. N. Rao, D. Lentz, H.-U. Reißig* Synthesis of Polycyclic Tertiary Carbinamines by Samarium Diiodide Mediated Cyclizations of Indolyl Sulfinyl Imines Angew. Chem. Int. Ed. 2015, 54, 2750 – 2753.
•	M. Kandziora, H.-U. Reißig* Synthesis of Rigid p-Terphenyl-Linked Carbohydrate Mimetics Beilstein J. Org. Chem. 2014, 10, 1749 – 1758.
•	C. Beemelmanns, S. Gross, H.-U. Reißig* *Towards the Core Structure of Strychnos* Alkaloids Using Samarium Diiodide-Induced Reactions of Indole Derivatives** Chem. Eur. J. 2013,19, 17801 – 17808.
•	A. Niermann, J. E. Grössel, H.-U. Reißig* New Thiochromans via Reductive Cyclization of Thiophenol Derivatives Synlett 2013, 177 – 180.
•	M. Jasiński,T. Watanabe, H.-U. Reißig* Samarium Diiodide Promoted Reduction of 3,6-Dihydro-2H-1,2-oxazines: Competition of 1,4-Amino Alcohol Formation and Ring Contraction to Pyrrole Derivatives Eur. J. Org. Chem. 2013, 605 – 610.
•	M. Berndt, A. Hölemann, A. Niermann, C. Bentz, R. Zimmer, H.-U. Reißig* Replacement of HMPA in Samarium Diiodide Promoted Cyclizations and Reactions of Organolithium Compounds Eur. J. Org. Chem. 2012, 1299 – 1302.
•	C. Beemelmanns, D. Lentz, H.-U. Reißig* Samarium Diiodide Induced Cyclizations of γ-, δ- and ε-Indolyl Ketones: Reductive Coupling, Intermolecular Trapping, and Subsequent Transformations of Indolines Chem. Eur. J. 2011, 17, 9720 – 9730.
•	C. Beemelmanns, H.-U. Reißig* Samarium diiodide induced ketyl-(het)arene cyclisations towards novel N-heterocycles Chem. Soc. Rev. 2011, 40, 2199 – 2210.
•	A. Niermann, H.-U. Reißig* Influence of Geminal Disubstitution on Samarium Diiodide Induced Reductive Cyclizatons of γ-Aryl Ketones Synlett 2011, 525 – 528.
•	C. Beemelmanns, H.-U. Reißig* New Samarium Diiodide-Induced Cyclizations Pure Appl. Chem. 2011, 83, 507 – 517.
•	J. Saadi, I. Brüdgam, H.-U. Reißig* Highly Substituted Benzannulated Cyclooctanol Derivatives by Samarium Diiodide-Induced Cyclizations Beilstein Journal of Organic Chemistry 2010, 6, No. 141, (1229 – 1245).
•	C. Beemelmanns, H.-U. Reißig* Eine kurze formale Strychnin-Totalsynthese mit einer Samariumdiiodid-induzierten Kaskadenreaktion als Schlüsselschritt Angew. Chem. 2010, 122, 8195 – 8199. C. Beemelmanns, H.-U. Reißig* A Short Formal Total Synthesis of Strychnine with a Samarium Diiodide Induced Cascade Reaction as the Key Step Angew. Chem. Int. Ed. 2010, 49, 8021 – 8025.
•	U. K. Wefelscheid, H.-U. Reißig* Synthesis of New Steroid Analogues by Samarium Diiodide Induced Cyclisations of γ-Naphthyl 1,3-Diones Tetrahedron: Asymmetry 2010, 21, 1601 – 1610.
•	C. Beemelmanns, V. Blot, S. Gross, D. Lentz, H.-U. Reißig* Highly Diastereoselective Samarium Diiodide Induced Ketyl Cyclisations of Indole and Pyrrole Derivatives – Scope and Limitations Eur. J. Org. Chem. 2010, 2716 – 2732.
•	C. Beemelmanns, H.-U. Reißig* Highly diastereoselective samarium diiodide induced cyclizations of new 3-substituted indole derivatives Org. Biomol. Chem. 2009, 7, 4475 - 4480.
•	J. Saadi, H.-U. Reißig* Scope and Limitations of Samarium Diiodide Induced Cyclizations of Alkenyl-Substituted γ-Keto Esters to Benzannulated Cyclooctanol Derivatives Synlett 2009, 2089 - 2092.
•	J. Saadi, D. Lentz, H.-U. Reißig* Medium-Sized Carbocycles by Samarium Diiodide-Induced Carbonyl-Alkene Cyclizations Org. Lett. 2009, 11, 3334 - 3337.
•	U. K. Wefelscheid, M. Berndt, H.-U. Reißig* Samarium Diiodide Mediated Ketyl-Aryl Couplings – Influence of Substituents and Trapping Experiments Eur. J. Org. Chem. 2008, 3635– 3646.
•	R. S. Kumaran, I. Brüdgam, H.-U. Reißig* Modular and Stereoselective Synthesis of Hydroxylated Angularly Fused Tricyclic Piperidine Derivatives via Samarium Diiodide-Mediated Cyclization Synlett, 2008, 991 – 994.
•	F. Aulenta, U. K. Wefelscheid, I. Brüdgam, H.-U. Reißig* Nitrogen-Containing Tricyclic and Tetracyclic Compounds via Stereoselective Samarium Diiodide Promoted Cyclizations of Quinolyl-Substituted Ketones – A New Access to Azasteroids Eur. J. Org. Chem. 2008, 2325 - 2335.
•	U. K. Wefelscheid, H.-U. Reißig* Pentacyclic Compounds by Samarium Diiodide-Induced Cascade Cyclizations of Naphthyl-Substituted 1,3-Diones Adv. Synth. Catal, 2008, 350, 65 – 69.
•	U. K. Wefelscheid, I. Brüdgam, H. Hartl, H.-U. Reißig* Crystal structure of (8S,9S,13S,14R,17S)-estra-1(10),2,4,6-tetraene- 14,17-diol monohydrate, C₁₈H₂₂O₂ H₂O Z. Kristallogr. NCS* 2007, 222, 467 – 468.
•	U. K. Wefelscheid, I. Brüdgam, H.-U. Reißig* Crystal structure of (8S,9S,13R,14R,17S)-9,17-cycloestra-1(10), 2,4,6-tetraene-14,17-diol trihydrate, C₁₈H₂₀O₂3H₂O Z. Kristallogr. NCS* 2007, 222, 465 – 466.
•	F. Aulenta, M. Berndt, I. Brüdgam, H. Hartl, S. Sörgel, H.-U. Reißig* A New, Efficient and Stereoselective Synthesis of Tricyclic and Tetracyclic Compounds by Samarium Diiodide Induced Cyclisations of Naphthyl-Substituted Arylketones – An Easy Access to Steroid-Like Skeletons Chem. Eur. J. 2007, 13, 6047 – 6062.
•	V. Blot, H.-U. Reißig* Efficient Synthesis of Medium-Sized Rings Incorporating Indole or Pyrrole Units by Samarium Diiodide Induced Cyclizations Eur. J. Org. Chem. 2006, 4989 - 4992.
•	F. Aulenta, H.-U. Reißig Heck Reactions of Quinoline-Derived Nonaflates Synlett 2006, 2993 – 2996.
•	V. Blot, H.-U. Reißig* Highly Substituted Dihydroindole Derivatives by Intermolecular Couplings of Samarium Ketyls and Indoles Synlett 2006, 2763 - 2766.
•	H.-U. Reißig, F. A. Khan, R. Czerwonka, C. U. Dinesh, A. L. Shaikh, R. Zimmer Benzannulated Cyclooctanol Derivatives by Samarium Diiodide Induced Intramolecular Carbonyl-Alkene Coupling - Scope, Limitations, Stereoselectivity Eur. J. Org. Chem.* 2006, 4419 - 4428.
•	F. Aulenta, A. Hölemann, H.-U. Reißig* Samarium Diiodide Induced Reactions of Cyclopropyl Ketones: Reductive Ring Cleavage and Dimerization Leading to 1,8-Diketones - Scope, Limitations, Mechanism Eur. J. Org. Chem. 2006, 1733 - 1739.
•	A. Hölemann, H.-U. Reißig* Samarium Diiodide in the Synthesis of Medium-Sized Rings - Carbocycles and Heterocycles by Intramolecular Addition of Samarium Ketyls to Alkynes Synlett 2004, 2732 - 2735.
•	A. Hölemann, H.-U. Reißig* Regioselective Samarium Diiodide-Induced Couplings of Carbonyl Compounds with 1,3-Diphenylallene and Alkoxyallenes - A New Route to 4-Hydroxy 1-Enol Ethers Chem. Eur. J. 2004, 10, 5493 - 5506.
•	A. Hölemann, H.-U. Reißig* Synthesis of New Furan Derivatives and 4-Hydroxy Aldehydes from 4-Hydroxy 1-Enol Ethers Synthesis 2004, 1963 – 1970.
•	M. Berndt, I. Hlobilová, H.-U. Reißig* Stereoselective Formation of Tri- and Tetracycles by Samarium Diiodide- Induced Cyclizations of Naphthyl-Substituted Ketones Org. Lett. 2004, 6, 957 - 960.
•	A. Hölemann, I. Brüdgam, H. Hartl, H.-U. Reißig Crystal Structure of cis-(5E)-Phenylmethylidenedecahydro-4aH-benzo[a]cyclo- hepten-4a-ol, C₁₈H₂₄O Z. Kristallogr. NCS* 2004, 219, 59 - 60.
•	S. Groß, I. Brüdgam, H. Hartl, H.-U. Reißig Crystal Structure of (9aRS,10SR,10aRS)-8-Methoxy-10-methyl- 1,2,3,5,7,9a,10,10a-octahydropyrrolo[1,2-b]isoquinoline-10-ol, C₁₄H₂₁NO₂ Z. Kristallogr. NCS* 2004, 219, 57 - 58.
•	S. Groß, I. Brüdgam, H. Hartl, H.-U. Reißig Crystal Structure of (4SR,4aSR)-1-Acetyl-4-hydroxy-4,8-dimethyl-1,2,3,4,4a,7- hexahydroquinoline, C₁₃H₁₉NO₂ Z. Kristallogr. NCS* 2004, 219, 55 - 56.
•	S. Groß, I. Brüdgam, H. Hartl, H.-U. Reißig Crystal Structure of (2RS,4SR,4aSR)-1-Acetyl-2-(1-methylethyl)-4-hydroxy- 4-methyl-1,2,3,4,4a,7-hexahydroquinoline, C₁₅H₂₂NO₂ Z. Kristallogr. NCS* 2004, 219, 53 - 54.
•	M. Berndt, I. Brüdgam, H. Hartl, H.-U. Reißig Crystal Structure of 1-Isopropyl-15-oxatetracyclo[11.2.1.02,11.05,10]hexadeca- 3,5(10),6,8-tetraen-14-one, C₁₈H₂₀O₂ Z. Kristallogr. NCS* 2004, 219, 51 - 52.
•	M. Berndt, I. Brüdgam, H. Hartl, H.-U. Reißig Crystal Structure of (1aSR,5bRS,7aSR,10aRS,10bSR,10cRS)-1a,5b,6,7,7a,8,9,10, 10b,10c-Decahydro-10aH-cyclopenta[1,2]phenanthro[9,10-b] oxiren-10a-ol, C₁₇H₂₀O₂ Z. Kristallogr. NCS* 2004, 219, 49 - 50.
•	M. Berndt, I. Brüdgam, H. Hartl, H.-U. Reißig Crystal Structure of (2SR,1'RS)-3-(1-Naphthyl)-2-(2-oxocyclopentyl)-propionic acid methyl ester, C₁₉H₂₀O₃ Z. Kristallogr. NCS* 2004, 219, 47 - 48.
•	M. Berndt, S. Groß, A. Hölemann, H.-U. Reißig* New Samarium Diiodide-Induced Ketyl Couplings – From Analogous Reactions to Serendipitously Discovered Processes Synlett 2004, 422 – 438.
•	S. Groß, H.-U. Reißig* Novel Stereoselective Syntheses of Highly Functionalized Benzannulated Pyrrolizidines and Indolizidines by Samarium Diiodide-Induced Cyclizations of Indole Derivatives Org. Lett. 2003, 5, 4305 - 4307.
•	A. Hölemann, H.-U. Reißig* Samarium Diiodide-Induced Couplings of Carbonyl Compounds with Methoxyallene Leading to 4-Hydroxy 1-Enol Ethers Org. Lett. 2003, 5, 1463 - 1466.
•	S. Groß, H.-U. Reißig* Samarium Diiodide-Induced Diastereoselective Synthesis of Hexahydroquinoline Derivatives Synlett 2002, 2027 - 2030.
•	O. Rademacher, R. Zimmer, C. U. Dinesh, H. U. Reißig Crystal structure of 2SR,5SR,5aSR,11bSR-5-Methyl-1,5,5a,11b- tetrahydro-2,5-methanonaphtho[2,1-c]oxepin-3(2H)-one, C₁₆H₁₆O₂ Z. Kristallogr. NCS* 2002, 217, 425 - 426.
•	O. Rademacher, R. Zimmer, C. U. Dinesh, H. U. Reißig Crystal structure of Methyl 4aSR,5RS,12aRS-12a-Hydroxy- 1,2-3,4,4a,5,6,11,12,12a-decahydro-dibenzo[a,e][8]annulene-5-carboxylate, C₁₈H₂₄O₃ Z. Kristallogr. NCS* 2002, 217, 423 - 424.
•	O. Rademacher, M. Berndt, H.-U. Reißig Crystal Structure of 4R,4aS,5S-5-Hydroxy-4-(1-hydroxy-1-methylethyl)-5- methyl-4,4a,5,6,7,8-hexahydronaphthalene-2-carbonitrile—water (1/1), C₁₅H₂₁NO₂ H₂O. Kristallogr. NCS 2001, 216, 593 – 594.
•	D. Lentz, E. Nandanan, H.-U. Reißig Crystal Structure of 6S,8S-9-Butyl-8-hydroxy-8-isopropyl-5,6,7,8-tetra hydrobenzocyclooctene-6-carboxylate, C₂₁H₃₀NO₃Z. Kristallogr.* NCS 2001, 216, 525 – 526.
•	Berndt, H.-U. Reißig* Substituent Effects in Samarium Diiodide-Induced 6-trig Cyclizations of γ-Aryl ketones to Functionalized Hexahydronaphthalene Derivatives Synlett 2001, 1290 – 1292.
•	C. U. Dinesh, H.-U. Reißig, O. Rademacher* Crystal structure of methyl 4aR,4bR,8aS,9R-1-cyano-4b-hydroxy-2,4a, 4b,5,6,7,8,8a,9, 10-decahydro- phenanthrene-9-carboxylate, C₁₇H₂₁NO₃ Z. Kristallogr. NCS 2000, 215, 615 - 616.
•	E. Nandanan, C. U. Dinesh, H.-U. Reißig* Competition between Novel 8-endo-dig and 6-trig Cyclizations of Samarium Ketyls Leading either to Benzannulated Cyclooctene or to Hexahydronaphthalene Derivatives Tetrahedron 2000, 56, 4267 - 4277.
•	R. Zimmer, G. Zahn, F. A. Khan, H.-U. Reißig Configurational Analysis of 14,14-Dimethyl-12-oxatricyclo[9.2.1.0^3,8]tetradeca- 3,5,7-trien-13-one Acta Crystallogr. Sect. C 1999, 55, 1941 - 1943.
•	C. U. Dinesh, H.-U. Reißig* Eine neue Samariumdiiodid-induzierte Reaktion: intramolekularer Angriff von Ketylradikalanionen auf Arylsubstituenten unter Bildung von 1,4-Cyclohexadienderivaten Angew. Chem. 1999, 111, 874 - 876.
	C. U. Dinesh, H.-U. Reißig* A New Samarium Diiodide Induced Reaction: Intramolecular Attack of Ketyl Radical Anions on Aryl Substituents with Formation of 1,4-Cyclohexadiene Derivatives Angew. Chem. Int. Ed. 1999, 38, 789 - 791.
•	F. A. Khan, R. Czerwonka, R. Zimmer, H.-U. Reißig* A Novel Sm(II)-Induced Route to Highly Substituted Benzannulated Cyclooctanol Derivatives Synlett 1997, 995 - 997.

Synthesis of Carbohydrates and Carbohydrate Mimetics

Publications

•	M. Jasiński, G. Utecht, A. Fruziński, H.-U. Reißig Three-Step Synthesis of 3-Aminoseptanoside Derivatives Using Lithiated Methoxyallene and δ-Siloxynitrones* Synthesis 2016, 48, 893 – 905.
•	J. Salta, J. Dernedde, H.-U. Reißig* Synthesis of Multivalent Carbohydrate Mimetics with Aminopolyol End Groups and their Evaluation as L-Selectin Inhibitors Beilstein J. Org. Chem. 2015, 11, 638 – 646.
•	J. Salta, H.-U. Reißig* Synthesis of Divalent Carbohydrate Mimetics by Reductive Amination with Enantiopure 1,2-Oxazines as Precursors Synthesis 2015, 47, 1893 – 1898.
•	M. Kandziora, E. Mucha, S. P. Zucker, H.-U.Reißig* Syntheses of Mono- and Divalent C-Aminoglycosides Using 1,2-Oxazine Chemistry and Olefin Metathesis Synlett 2015, 26, 367 – 374.
•	M. Kandziora, H.-U. Reißig* Preparation of Multivalent Carbohydrate Mimetics Based on Enantiopure 1,2-Oxazines by Sonogashira Coupling and Subsequent Reductive Ring-Opening Eur. J. Org. Chem. 2015, 370 – 377.
•	L. Bouché, M. Kandziora, H.-U. Reißig* Synthesis of New Enantiopure Poly(hydroxy)aminooxepanes as Building Blocks for Multivalent Carbohydrate Mimetics Beilstein J. Org. Chem. 2014, 10, 213 – 223.
•	M. Jasiński, Dieter Lentz, E. Moreno-Clavijo, H.-U. Reißig* Application of L-Erythrose-Derived Nitrones in the Synthesis of Polyhydroxylated Compounds via 3,6-Dihydro-2H-1,2-oxazine Derivatives Eur. J. Org. Chem. 2012, 3304 – 3316.
•	M. Jasiński, Dieter Lentz, H.-U. Reißig* Carbohydrate-Auxiliary Assisted Preparation of Enantiopure 1,2-Oxazine Derivatives and Aminopolyols Beilstein J. Org. Chem. 2012, 8, 662-674.
•	L. Bouché, H.-U. Reißig* Synthesis of Novel Carbohydrate Mimetics via 1,2-Oxazines Pure Appl. Chem. 2012, 84, 23 – 36.
•	M. Roskamp, S. Enders, F. Pfrengle, S. Yekta. V. Dekaris, J. Dernedde, H.-U. Reißig, S. Schlecht* Multivalent Interaction and Selectivities in Selectin Binding of Functionalized Gold Colloids Decorated with Carbohydrate Mimetics Org. Biomol. Chem. 2011, 9, 7448 – 7456.
•	V. Dekaris, R. Pulz, A. Al-Harrasi, D. Lentz, H.-U. Reißig* Stereoselective Synthesis of Aza, Amino and Imion Sugar Derivatives by Hydroboration of 3,6-Dihydro-2H-1,2-oxazines as Key Reaction Eur. J. Org. Chem. 2011, 3210 – 3219.
•	G. Semini, A. Hildmann, H.-U. Reißig, W. Reutter, K. Danker* The Novel Synthetic Ether Lipid Inositol-C2-PAF Inhibits Phosphorylation of the Tyrosine Kinases Src and FAK Independent of Integrin Activation in Transformed Skin Cells Biochemical Pharmacology 2011, 81, 985 – 995.
•	A. Al-Harrasi, L. Bouché, R. Zimmer, H.-U. Reißig* β-Alkoxy-γ-amino Aldehydes by Internal Redox Ring Cleavages of Carbohydrate-Derived Enantiopure 1,2-Oxazines and Preparation of Heterocycles with Aminopolyol Side Chain Synthesis 2011, 109 – 118.
•	F. Pfrengle, H.-U. Reißig* Internally Protected Amino Sugar Equivalents from Enantiopure 1,2-Oxazines: Synthesis of Variably Configured Carbohydrates with C-Branched Amino Sugar Units Chem. Eur. J. 2010, 16, 11915 – 11925.
•	F. Pfrengle, H.-U. Reißig* Addition of Lithiated Enol Ethers to Nitrones and Subsequent Lewis Acid Induced Cyclizations to Enantiopure 3,6-Dihydro-2H-pyrans – an Approach to Carbohydrate Mimetics Beilstein Journal of Organic Chemistry 2010, 6, No. 75.
•	F. Pfrengle, H.-U. Reißig* *Amino Sugars and their Mimetics via* 1,2-Oxazines** Chem. Soc. Rev., 2010, 39, 549 – 557.
•	A. Al-Harrasi, S. Fischer, R. Zimmer, H.-U. Reißig* Ring Enlargement of Carbohydrate-Derived 1,2-Oxazines to Enantiopure 5-Bromo-1,2-oxazepines and Subsequent Palladium-Catalyzed Reactions Synthesis 2010, 304 – 314.
•	V. Dekaris, B. Bressel, H.-U. Reißig* Acid Mediated Transformations of Enantiopure 3,6-Dihydro-2H-1,2-oxazines into Functionalized Aminotetrahydrofuran Derivatives Synlett 2010, 47 – 50.
•	V. Dekaris, H.-U. Reißig* Stereocontrolled Syntheses of Enantiopure Polyhydroxylated Azetidines via 1,2-Oxazines Synlett 2010, 42 – 46.
•	F. Pfrengle, D. Lentz, H.-U. Reißig* A New Ring Closure Approach to Enantiopure 3,6-Dihydro-2H-pyrans: Stereodivergent Access to Carbohydrate Mimetics Org. Lett. 2009, 11, 5534 – 5537.
•	A. Al-Harrasi, F. Pfrengle, V. Prisyazhnyuk, S. Yekta, P. Koóš, H.-U. Reißig* Enantiopure Aminopyrans by a Lewis Acid Promoted Rearrangement of 1,2-Oxazines: Versatile Building Blocks for Oligosaccharide and Sugar Amino Acid Mimetics Chem. Eur. J. 2009, 15, 11632 – 11642
•	M. Brasholz, H.-U. Reißig* Alkoxyallene-Based De Novo Synthesis of Rare Deoxy Sugars: New Routes to L-Cymarose, L-Sarmentose, L-Diginose and L-Oleandrose Eur. J. Org. Chem. 2009, 3595– 3604.
•	F. Pfrengle, D. Lentz, H.-U. Reißig* Stereodivergente De-novo-Synthese verzweigter Aminozucker durch Lewis-Säure-induzierte Umlagerung von 1,2-Oxazinen Angew. Chem. 2009, 121, 3211 - 3215.
	F. Pfrengle, D. Lentz, H.-U. Reißig* Stereodivergent De novo Synthesis of Branched Amino Sugars by Lewis Acid promoted Rearrangement of 1,2-Oxazines Angew. Chem. Int. Ed. 2009, 48, 3165 - 3169.
•	B. Bressel, H.-U. Reißig* A New Approach to Neuraminic Acid Analogues via 1,2-Oxazines Org. Lett. 2009, 11, 527 – 530.
•	F. Pfrengle, A. Al-Harrasi, I. Brüdgam, H.-U. Reißig* Unusual Enantiopure Heterocyclic Skeletons via Lewis Acid Promoted Rearrangements of 1,3-Dioxolanyl-Substituted 1,2-Oxazines Eur. J. Org. Chem. 2009, 282 – 291.
•	E. Hýrošovà, L. Fišera,* M. Medvecký, H.-U. Reißig, A. Al-Harrasi, M. Koòš From sugars to modified nucleosides ARKIVOC 2009 (ix), 122 - 142.
•	B. Bressel, B. Egart, A. Al-Harrasi, R. Pulz, H.-U. Reißig,* I. Brüdgam Acid-Induced and Reductive Transformations of Enantiopure 3,6-Dihydro-2H-1,2-oxazines – Synthesis of Dideoxyamino Carbohydrate Derivatives Eur. J. Org. Chem. 2008, 467 – 474.
•	S. Yekta, V. Prisyazhnyuk, H.-U. Reißig* Simple Modifications of Enantiopure 1,2-Oxazines Leading to Building Blocks for Carbohydrate and Peptide Mimetics Synlett 2007, 2069 – 2072.
•	M. Brasholz, H.-U. Reißig* Oxidative Spaltung von 3-Alkoxy-2,5-dihydrofuranen und ihre Anwendung in der De-novo-Synthese seltener Monosaccharide am Beispiel von L-Cymarose Angew. Chem. 2007, 119, 1659 – 1662; Angew. Chem. Int. Ed. 2007, 46, 1634 – 1637.
•	A. Al-Harrasi, I. Brüdgam, H. Hartl, H.-U. Reißig* Crystal structure of 1R,5S,8R,9S-8-azidomethyl-2-benzyl- 6,6-dimethyl-3,7-dioxa-2-aza-bicyclo[3.3.1]nonan-9-0l, C₁₆H₂₂N₄O₃ Z. Kristallogr. NCS 2005, 220, 599 - 600.
•	A. Al-Harrasi, I. Brüdgam, H. Hartl, H.-U. Reißig* Crystal structure of 3S,4S,5R,6S,7R-5-amino-6-(tert-butyldimethylsiloxy)- 7(tert-butyldimethylsiloxymethyl)-3-hydroxymethyl-2,2-dimethyloxepan-4-ol, C₂₂H₄₉NO₅Si₂Z. Kristallogr. NCS 2006, 221, 131 – 132.
•	A. Al-Harrasi, H.-U. Reißig* Enantiomerenreiner Kohlenhydratmimetika durch Lewis-Säure-induzierte Umlagerung von 1,3-dioxolanyl-substitutierten 3,6-Dihydro-2H-1,2-oxazinen Angew. Chem. 2005, 117, 6383 - 6387.
•	A. Al-Harrasi, H.-U. Reißig* Synthesis of Enantiopure Carbohydrate Mimetics by Lewis Acid Catalyzed Rearrangement of 1,3-Dioxolanyl-Substituted 1,2-Oxazines Angew. Chem. Int. Ed. 2005, 44, 6227 – 6231.
•	A. Al-Harrasi, H.-U. Reißig* Synthesis of Enantiopure Functionalized β-Alkoxy γ-Amino Aldehydes by a New Internal Redox Ring Cleavage of Carbohydrate Derived 1,2-Oxazines Synlett 2005, 1152 – 1154.
•	R. Pulz, A. Al-Harrasi, H.-U. Reißig* Acid Promoted Syntheses of New Enantiopure Amino Sugar Derivatives from 3,6-Dihydro-2H-1,2-oxazines Synlett 2002, 817 – 819.

Multicomponent Reactions with Donor-Acceptor-Substituted Cyclopropanes

Publications

•	J. Saadi, C. Bentz, K. Redies, D. Lentz, R. Zimmer, H.-U. Reißig* Stereoselective Synthesis of Tricyclic Compounds by Intramolecular Palladium-Catalyzed Addition of Aryl Iodides to Carbonyl Groups Beilstein J. Org. Chem. 2016, 12, 1236 – 1242.
•	D. Reich, D. S. Müller, L. Schefzig, R. Zimmer,* H.-U. Reißig* One-Pot Generation of C≡X Bonds from Methyl 2-Siloxycyclopropanecarboxylates: Simple Syntheses of Functionalized Nitriles and Alkynes Synlett 2014, 25, 2265 – 2270.
•	T. H. Ngo, H. Berndt, M. Wilsdorf, D. Lentz, H.-U. Reißig* Linear and Cyclic Hybrids of Alternating Thiophene–Amino Acid Units: Synthesis and Effects of Chirality on Conformation and Molecular Packing Chem. Eur. J. 2013,19, 15155 – 15165.
•	D.Gladow, H.-U. Reißig* Alkylation and Ring Opening of Perfluoroalkyl- and Perfluoroaryl-Substituted 2-Siloxycyclopropanecarboxylates Yielding Fluorinated γ-Oxo Esters or β,γ-Unsaturated Ketones Synthesis 2013, 2179 – 2187.
•	M. H. Beyzavi, C. Nietzold, H.-U. Reißig, A. Wiehe Synthesis of Functionalized trans-A2B2-Porphyrins Using Donor-Acceptor Cyclopropane-Derived Dipyrromethanes Adv. Synth. Catal. 2013, 355, 1409 – 1422.
•	M. H. Beyzavi, D. Lentz, H.-U. Reißig, A. Wiehe Synthesis of New Functionalized Calix[n]phyrin Macrocycles with Varied Ring Sizes by Using a Sterically Congested Dipyrromethane Chem. Eur. J. 2013, 19, 6203 – 6208.
•	M. H. Beyzavi, D. Lentz, H.-U. Reißig, A. Wiehe Synthesis of Functionalized, Sterically Congested Calix[4]phyrin Macrocycles Using Donor-Acceptor-Substituted Cyclopropanes – First Example of a Mono-meso-spirolactone Incorporated into a Calix[4]phyrin Eur. J. Org. Chem. 2013, 269 – 282.
•	T. H. Ngo, H. Berndt, D. Lentz, H.-U. Reißig* Linear and Cyclic Amides with a Thiophene Backbone: Ultrasound-Promoted Synthesis and Crystal Structures J. Org. Chem. 2012, 77, 9676 – 9683.
•	D. Gladow, H.-U. Reißig* Synthesis of Perfluoroalkyl-Substituted γ-Lactones and 4,5-Dihydropyridazin-3(2H)-ones via Donor-Acceptor Cyclopropanes Helv. Chim. Acta 2012, 95, 1818 – 1830.
•	H. A. Laub, D. Gladow, H.-U. Reißig, H. Mayr The Influence of Perfluorinated Substitutents on the Nucleophilic Reactivities of Silyl Enol Ethers Org. Lett. 2012, 14, 3990 – 3993.
•	H. Özbek, D. Lentz, H.-U. Reißig* New Macrocyclic Peptidomimetics Containing 5-Aminothiophene Subunits Eur. J. Org. Chem. 2010, 6319 – 6322.
•	H. Özbek, I. S. Veljkovic, H.-U. Reißig* Gewald Synthesis of Aminothiophene Carboxylic Acids Providing New Dipeptide Analogues Synlett 2008, 3145 – 3148.
•	I. Veljkovic, R. Zimmer, H.-U. Reißig, I. Brüdgam, H. Hartl A Flexible Three-Component Synthesis of Novel δ-Amino Acids Incorporating an Imidazo[1,2-α]pyridine Backbone* Synthesis 2006, 2677 - 2684.
•	R. Zimmer, A. Ziemer, M. Gruner, I. Brüdgam, H. Hartl, H.-U. Reißig* Siloxycyclopropanes in Ugi Four-Component Reaction: A New Method for Synthesis of Highly Substituted Pyrrolidinone Derivatives Synthesis 2001, 1649 - 1658.

Cross Coupling Reactions of Alkenyl Nonaflates

Publications

•	M. Taszarek, H.-U. Reißig* Heck Reactions and Carbonylations of Alkenyl Nonaflates – Synthesis of Tetradehydroamino Acids and α,β-Unsaturated Carboxylic Acids ChemistrySelect 2016, 1, 5712 – 5715.
•	P. Hommes, H.-U. Reißig* Synthesis of Highly Functionalized 2,2´-Bipyridines by Cyclocondensation of β-Ketoenamides – Scope and Limitations Beilstein J. Org. Chem. 2016, 12, 1170 – 1177.
•	G. Podolan, L. Hettmanczyk, P. Hommes, B. Sarkar,* H.-U. Reißig* Synthesis and (Spectro)electrochemistry of New Ferrocenyl-Substituted Pyridine Derivatives Eur. J. Org. Chem. 2015, 7317 – 7323.
•	J. Högermeier, D. Trawny, R. Zimmer, H.-U. Reissig* Diels-Alder Reactions of 1,3-Dienes Incorporated into 8-Oxa- and 8-Thia-bicyclo[3.2.1]octane Skeletons: A Convenient Access to Complex Tri- and Tetracyclic Compounds Synthesis 2015, 47, 2767 – 2775.
•	D. Trawny, M. Quennet, N. Rades, D. Lentz, B. Paulus, H.-U. Reissig* Syntheses, Structures and Conformational Dynamics of 1,3,5-Tris(3‘‘-ethynylbi-phenyl-2‘-yl)benzene Derivatives Eur. J. Org. Chem. 2015, 4667 – 4674.
•	J. Dash, D. Trawny, J. P. Rabe, H.-U. Reissig* C₃-Symmetric Pyridine and Bipyridine Derivatives: Simple Preparation by Cyclocondensation and 2D Self-Assembly at a Solution-Graphite Interface Synlett 2015, 26, 1486 – 1489.
•	D. Trawny, V. Kunz, H.-U. Reißig* Modular Syntheses of Star-Shaped Pyridine, Bipyridine, and Terpyridine Derivatives by Employing Sonogashira Reactions Eur. J. Org. Chem. 2014, 6295 – 6302.
•	D. Gladow, S. Doniz-Kettenmann, H.-U. Reißig* 1,3-Dipolar Cycloadditions of Ethyl 2-Diazo-3,3,3-trifluoropropanoate to Alkynes and [1,5] Sigmatropic Rearrangements of the Resulting 3H-Pyrazoles: Synthesis of Mono-, Bis- and Tris(trifluoromethyl)-Substituted Pyrazoles Helv. Chim. Acta, 2014, 97, 808 – 821.
•	D. Gladow, H.-U. Reißig* Perfluoroalkyl-Substituted Thiophenes and Pyrroles from Donor-Acceptor Cyclopropanes and Heterocumulenes: Synthesis and Exploration of their Reactivity J. Org. Chem. 2014, 79, 4492 – 4502.
•	L. Bouché, H.-U. Reißig* Synthesis of Di- and Trivalent Carbohydrate Mimetics with Oxepane Substructure by Employing Copper-Catalyzed [3+2] Cycloadditions of Alkynes with Azidooxepanes Eur. J. Org. Chem. *2014,* 3697 – 3703.
•	M. Domínguez, H.-U. Reißig* New 4-Pyridyl Nonaflates as Precursors for Push-Pull Solvatochromik Dyes Synthesis 2014, 46, 1110 – 1106.
•	M. K. Bera, M. Domínguez, P. Hommes, H.-U. Reißig* The Flögel-Three-Component Reaction with Dicarboxylic Acids - An Approach to Bis(β-alkoxy-β - ketoenamides) for the Synthesis of Complex Pyridine and Pyrimidine Derivatives Beilstein J. Org. Chem. 2014, 10, 394 – 404.
•	M. K. Bera, S. L. Gholap, P. Hommes, K. Neuthe, D. Trawny, J. P. Rabe, D. Lentz, R. Zimmer, H.-U. Reißig* Synthesis and Properties of Branched Oligo(2-thienyl)- and Oligo(2,2’-bithien-5-yl)-Substituted Pyridine Derivatives Adv. Synth. Catal. 2013, 355, 3463 – 3474
•	P. Hommes, S. Berlin, H.-U. Reißig* Trimethylsilyl Trifluoromethanesulfonate-Promoted Cyclocondensation of b-Keto-enamides and Subsequent Nonaflation to Pyrid-2-yl and Pyrid-4-yl Nonaflates as Flexible Precursors for Polysubstituted Pyridines Synthesis 2013, 45, 3288 – 3294.
•	S. L. Gholap, P. Hommes, K. Neuthe, H.-U. Reißig* Per(2-thienyl)pyridines: Synthesis and Properties Org. Lett. 2013, 15, 318 – 321.
•	T. Lechel, G. Podolan, B. Brusilowskij, C. A. Schalley, H.-U. Reißig* Unexpected One-Step Formation of Iodo[1,3]dioxolo[4,5-c]pyridine Derivatives by a Hofmann-Löffler-Freytag Reaction: Studies on the Synthesis of a Pyridine-Containing Macrocycle Eur. J. Org. Chem. 2012, 5685 – 5692.
•	C. Eidamshaus, P. Hommes, H.-U. Reißig* Palladium-Catalyzed Coupling of Pyrid-4-yl Nonaflates with Methyl Diazoacetate Synlett 2012, 1670 – 1674.
•	C. Eidamshaus, T. Triemer, H.-U. Reißig* *Synthesis of 4-Quinolones via Cyclocondensation of Substituted ortho-Amidoacetophenones: A Refit to the Camps Cyclization by Applying Trimethylsilyl Trifluoromethanesulfonate/Triethylamine* Synthesis 2011, 3261 – 3266.
•	C. Eidamshaus, H.-U. Reißig* A Chiral Pool Strategy for the Synthesis of Enantiopure Hydroxymethyl-Substituted Pyridine Derivatives Eur. J. Org. Chem. 2011, 6056 – 6069
•	M. K. Bera, P. Hommes, H.-U. Reißig* In Search of Oligo(2-thienyl)-Substituted Pyridine Derivatives: A Modular Approach to Di-, Tri- and Tetra(2-thienyl)pyridines Chem. Eur. J. 2011, 17, 11838 – 11844.
•	P. Hommes, P. Jungk, H.-U. Reißig* Four-Component Synthesis of Functionalized 2,2’-Bipyridines Based on the Blaise Reaction Synlett 2011, 2311 – 2314.
•	T. Lechel, J. Dash, C. Eidamshaus, I. Brüdgam, D. Lentz, H.-U. Reißig* A Three-component Synthesis of β-Alkoxy-β-keto-enamides - Flexible Precoursors for 4-Hydroxypyridine Derivatives and their Palladium-catalysed Reactions Org. Biomol. Chem. 2010, 8, 3007 – 3014.
•	T. Lechel, I. Brüdgam, H.-U. Reißig* Preparation of pyridine-3,4-diols, their crystal packing and their use as precursors for palladium-catalyzed cross-coupling reactions Beilstein Journal of Organic Chemistry 2010, 6, No. 42.
•	J. Högermeier, H.-U. Reißig* Nine Times Fluoride can be Good for your Syntheses. Not just Cheaper: Nonafluorobutanesulfonates as Intermediates for Transition Metal-Catalyzed Reactions Adv. Synth. Catal. 2009, 351, 2747 – 2763.
•	J. Högermeier, H.-U. Reißig* Mild and Efficient Sonogashira Couplings of 8-Oxa- and 8-Thiabicyclo[3.2.1]octanone Derived Alkenyl Nonaflates Tetrahedron 2007, 63, 8485 – 8491.
•	J. Högermeier, H.-U. Reißig* First Comprehensive Investigation of Suzuki Couplings of Alkenyl Nonaflates with Aryl and Alkenyl Boronic Acid Derivatives by Using Classical Conditions and Microwave Heating Chem. Eur. J. 2007, 13, 2410 – 2420.
•	F. Aulenta, H.-U. Reißig* Heck Reactions of Quinoline-Derived Nonaflates Synlett 2006, 2993 - 2996.
•	J. Högermeier, H.-U. Reißig* Suzuki Couplings of New Bicyclic Boronic Esters Derived from 8-Heterobicyclo[3.2.1]octenyl Nonaflates and Application to the Synthesis of an Epibatidine-Atropine Hybrid Synlett 2006, 2759 - 2762.
•	J. Högermeier, H.-U. Reißig, I. Brüdgam, H. Hartl Nonaflates from 8-Oxabicyclo[3.2.1]oct-6-en-3-ones as Building Blocks for Diversity Orientated Synthesis: Preparation, Heck-Couplings and Subsequent Diels-Alder Reactions* Adv. Synth. Catal. 2004, 346, 1868 – 1879.
•	I. M. Lyapkalo, J. Högermeier, H.-U. Reißig* Synthesis of New Tropinone Derivatives by Palladium-Catalyzed Couplings of 8-Azabicyclo[3.2.1]oct-2-enyl Nonaflates Tetrahedron 2004, 60, 7721 - 7729.
•	I. M. Lyapkalo, H. U. Reißig, A. Schäfer, A. Wagner Study of Unusually High Rotation Barriers about S,N Bonds in Nonafluoro-1-butanesulfonamides: Electronic Nature of the Torsional Effect* Helv. Chim. Acta 2002, 85, 4206 – 4215.
•	I. M. Lyapkalo, M. Webel, H.-U. Reißig* One-Pot Transformation of Silyl Enol Ethers into 1,3-Dienes: In Situ Generation of Alkenyl Nonaflates Followed by Heck Reactions – Scope and Limitations Eur. J. Org. Chem. 2002, 3646 – 3658.
•	I. M. Lyapkalo, M. Webel, H.-U. Reißig* An Expedient and Stereoselective Synthesis of Alkenyl Nonaflates from Silyl Enol Ethers: Optimization, Scope and Limitations Eur. J. Org. Chem. 2002, 1015 - 1025.
•	I. M. Lyapkalo, M. Webel, H.-U. Reißig* Synthesis and Heck Reactions of Ethenyl and (Z)-Butadien-1-yl Nonaflate Obtained by Fragmentation of Furan Derivatives Eur. J. Org. Chem. 2001, 4189 – 4194.
•	I. M. Lyapkalo, M. Webel, H.-U. Reißig* *Enantioselective Synthesis of Cyclohexenylalkenes by Asymmetric Deprotonation of 4-tert-Butylcyclohexanone Followed by O-Nonaflation and Heck Couplings* Synlett 2001, 1293 – 1295.
•	R. Zimmer, M. Webel, H.-U. Reißig Nonafluoro-1-butanesulfonyl Fluoride: More than a Fluorinating Reagent* J. Prakt. Chem. 1998, 340, 274 – 277.
•	M. Webel, H.-U. Reißig* Heck Reactions Starting from Silyl Enol Ethers - A Simple One-Pot Nonaflation-Coupling Procedure for the Synthesis of 1,3-Dienes Synlett 1997, 1141 – 1142.
•	E. Hirsch, S. Hünig, H.-U. Reißig Darstellung von Enolsulfonsäureestern aus Trimethylsilylenolethern: Synthetische Konsequenz eines bemerkenswerten Kationeneffekts* Chem. Ber. 1982, 115, 3687 – 3696.

Department of Biology, Chemistry, Pharmacy

The Reissig Research Group

Current Topics

Metalated Alkoxy Allenes as Building Blocks for Synthesis of Heterocycles

Publications

Synthesis of Natural Products and Analogues

Synthesis of Natural Products and Analogues

Publications

Synthesis of Novel Pyridine Derivatives

Publications

Samarium Diiodide Induced Cyclization Reactions

Publications

Synthesis of Carbohydrates and Carbohydrate Mimetics

Synthesis of Carbohydrates and Carbohydrate Mimetics

Publications

Multicomponent Reactions with Donor-Acceptor-Substituted Cyclopropanes

Publications

Cross Coupling Reactions of Alkenyl Nonaflates

Publications