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Kinetics, Thermodynamics, and Structural Effects of Quinoline-2-Carboxylates, Zinc-Binding Inhibitors of New Delhi Metallo-β-lactamase-1 Re-sensitizing Multidrug-Resistant Bacteria for Carbapenems

Jia Y.; Schroeder B.; Pfeifer Y.; Fröhlich C.; Deng L.; Arkona C.; Kuropka B.; Sticht J.; Ataka K.; Bergemann S.; Wolber G.; Nitsche C.; Mielke M.; Leiros H.S.; Werner G.; Rademann J. – 2023

Title
Kinetics, Thermodynamics, and Structural Effects of Quinoline-2-Carboxylates, Zinc-Binding Inhibitors of New Delhi Metallo-β-lactamase-1 Re-sensitizing Multidrug-Resistant Bacteria for Carbapenems
Author
Jia Y.; Schroeder B.; Pfeifer Y.; Fröhlich C.; Deng L.; Arkona C.; Kuropka B.; Sticht J.; Ataka K.; Bergemann S.; Wolber G.; Nitsche C.; Mielke M.; Leiros H.S.; Werner G.; Rademann J.
Date
2023
Source(s)
Appeared in
J. Med. Chem. 2023, 66, 11761–11791
Citation
DOI: 10.1021/acs.jmedchem.3c00171
Type
Text